SCHEMBL9255566

SCHEMBL9255566

CCOC(=O)c1[nH]c2ccc(C)cc2c1CNCCC1CCN(Cc2ccccc2)CC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 8/20 0.51
BCHE P06276 4/20 0.51
ALDH1A1 P00352 4/20 0.51
KDM4E B2RXH2 3/20 0.51
HPGD P15428 3/20 0.51
MAPT P10636 2/20 0.51
HSD17B10 Q99714 2/20 0.51
USP2 O75604 1/20 0.51
MAPK1 P28482 1/20 0.51
CASP7 P55210 1/20 0.51
MAOB P27338 4/20 0.51
MAOA P21397 2/20 0.51
DRD2 P14416 1/20 0.49
DRD4 P21917 1/20 0.49
DRD3 P35462 1/20 0.49
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
HIF1A Q16665 1/20 0.48
CNR1 P21554 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9260014 0.93 CNR1 (0.56) ACHEBCHEALDH1A1KDM4EHPGD
SCHEMBL9251113 0.91 ACHE (0.54) ACHEBCHEALDH1A1KDM4EHPGD
SCHEMBL9265225 0.86 ACHE (0.60) ACHEBCHEALDH1A1KDM4EHPGD
SCHEMBL9260634 0.84 ACHE (0.54) ACHEBCHEMAOBMAOA
SCHEMBL9255557 0.80 ALDH1A1 (0.50) ACHEBCHEALDH1A1KDM4EHPGD
SCHEMBL9251812 0.77 ACHE (0.64) ACHEBCHEMAOBMAOA
SCHEMBL9254634 0.75 MAOB (0.51) ACHEBCHEMAOBMAOA
SCHEMBL9261890 0.74 ACHE (0.51) ACHEBCHEMAOBMAOA
SCHEMBL9260006 0.73 CNR1 (0.53) ACHEBCHEALDH1A1KDM4EHPGD
SCHEMBL9251106 0.71 KDM4E (0.51) ACHEALDH1A1KDM4EHPGDMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5428043-A Tricyclic-cyclic amines as novel cholinesterase inhibitors PFIZER INC. (US) 1995-06-27 US disclosed
EP-0441517-A2 Tricyclic amines as novel cholinesterase inhibitors PFIZER INC. (US) 1991-08-14 EP disclosed