SCHEMBL9255518

SCHEMBL9255518

COC(=O)CCNC(=O)c1cc2nc(-c3ccc(C(=N)N)cc3)n(C)c2cc1OCCCc1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 1/20 0.41
RAB9A P51151 1/20 0.40
F10 P00742 1/20 0.40
HDAC1 Q13547 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
PTGES O14684 1/20 0.39
PRSS12 P56730 2/20 0.38
PDE4A P27815 3/20 0.38
PDE4B Q07343 3/20 0.38
PDE4C Q08493 3/20 0.38
PDE4D Q08499 3/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2B6 P20813 1/20 0.38
EHMT2 Q96KQ7 1/20 0.38
PLK1 P53350 1/20 0.38
TP53 P04637 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9254618 0.94 CHEK2 (0.42) CHEK2F10HDAC1HDAC8HDAC6
SCHEMBL9252426 0.89 PRSS12 (0.39) CHEK2F10HDAC1HDAC8HDAC6
SCHEMBL9255533 0.86 NPC1 (0.40) CHEK2RAB9AHDAC1HDAC8HDAC6
SCHEMBL9249762 0.84 ITGB3 (0.42) CHEK2F10HDAC1HDAC8HDAC6
SCHEMBL9255062 0.82 CHEK2 (0.40) CHEK2F10HDAC1HDAC8HDAC6
SCHEMBL9248606 0.82 EHMT2 (0.49) RAB9AF10EHMT2TP53
SCHEMBL9252912 0.82 ITGB3 (0.43) CHEK2HDAC1HDAC8HDAC6PRSS12
SCHEMBL9245485 0.82 PTGER4 (0.48) RAB9AF10CYP1A2CYP3A4CYP2D6
SCHEMBL9249905 0.81 CHEK2 (0.39) CHEK2RAB9AHDAC1HDAC8HDAC6
Acetic Acid SCHEMBL9256132 0.80 CHEK2 (0.39) CHEK2RAB9AF10HDAC1HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5434150-A Anticoagulants, cardiovascular disorders DR. KARL THOMAE GMBH (DE) 1995-07-18 US disclosed
EP-0531883-A1 Condensed 5-membered ring heterocycles, process for their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1993-03-17 EP disclosed