SCHEMBL9255571

SCHEMBL9255571

Cc1csc(Oc2ccc(-c3c(C)oc(C)cc3=O)cc2)c1

nearest known ligand 0.42

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 18/20 0.42
PTGS1 P23219 1/20 0.42
ACHE P22303 1/20 0.36
MAPT P10636 1/20 0.35
ATM Q13315 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9269944 0.79 EGFR (0.49) PTGS2PTGS1ACHEMAPTATM
SCHEMBL9264843 0.78 PTGS2 (0.52) PTGS2PTGS1ACHE
SCHEMBL9265538 0.78 PTGS2 (0.52) PTGS2PTGS1ACHE
SCHEMBL9256975 0.77 PTGS2 (0.60) PTGS2PTGS1
SCHEMBL9271420 0.77 MAPT (0.51) PTGS2MAPTATM
SCHEMBL9268153 0.77 PTGS2 (0.45) PTGS2PTGS1ACHE
SCHEMBL9255564 0.76 ACHE (0.41) PTGS2PTGS1ACHEMAPT
SCHEMBL9268345 0.75 PTGS2 (0.55) PTGS2PTGS1ACHEMAPT
SCHEMBL9266183 0.75 PTGS2 (0.55) PTGS2PTGS1ACHE
SCHEMBL9282952 0.75 PTGS2 (0.53) PTGS2PTGS1ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5403934-A Heterocyclic compounds BURROUGHS WELLCOME CO. (US) 1995-04-04 US disclosed
WO-1991013873-A1 HETEROCYCLIC COMPOUNDS THE WELLCOME FOUNDATION LIMITED (GB) 1991-09-19 WO disclosed
EP-0447164-A1 Heterocyclic compounds THE WELLCOME FOUNDATION LIMITED (GB) 1991-09-18 EP disclosed