SCHEMBL9255665

SCHEMBL9255665

CCOC(=O)c1cn(Cc2ccccc2)c(CO)n1

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.56
LMNA P02545 2/20 0.56
GABRA2 P47869 4/20 0.50
GABRB2 P47870 4/20 0.50
F2RL3 Q96RI0 1/20 0.49
KDM4E B2RXH2 1/20 0.47
CYP19A1 P11511 1/20 0.47
CYP1A2 P05177 1/20 0.47
CRHBP P24387 1/20 0.46
CRHR2 Q13324 1/20 0.46
MAPT P10636 2/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
MAPK1 P28482 2/20 0.46
GAA P10253 1/20 0.46
P2RX7 Q99572 1/20 0.46
TSHR P16473 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16862955 0.85 ALDH1A1 (0.60) ALDH1A1LMNAGABRA2GABRB2F2RL3
SCHEMBL9256717 0.80 BRD4 (0.52) ALDH1A1SMN1; SMN2GAAP2RX7TSHR
SCHEMBL31132944 0.79 ALDH1A1 (0.53) ALDH1A1LMNAGABRA2GABRB2F2RL3
SCHEMBL13437651 0.78 CYP19A1 (0.61) ALDH1A1LMNAGABRA2GABRB2F2RL3
SCHEMBL29339719 0.75 ALDH1A1 (0.53) ALDH1A1LMNAF2RL3KDM4ECYP19A1
SCHEMBL17241086 0.73 P2RX7 (0.46) ALDH1A1LMNAKDM4ECYP1A2SMN1; SMN2
SCHEMBL2117362 0.73 MAPK1 (0.52) ALDH1A1LMNAF2RL3KDM4ECYP19A1
SCHEMBL6801734 0.72 KDM4E (0.49) ALDH1A1LMNAGABRA2GABRB2KDM4E
SCHEMBL27094252 0.72 DGAT1 (0.45) ALDH1A1GABRA2GABRB2KDM4ECYP1A2
SCHEMBL9248509 0.72 LMNA (0.60) ALDH1A1LMNAGABRA2GABRB2CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5395838-A Aromatic aminomethyl substitutes compounds IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1995-03-07 US disclosed
EP-0373891-B1 Anti-tumour agents ICI PLC (GB) 1994-11-02 EP disclosed
US-5252573-A Quinazoline derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-10-12 US disclosed
US-5089499-A Anticarcinogenic agents; thymidylate synthetase inhibitors; antiallergens; psoriasis IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-02-18 US disclosed
EP-0373891-A2 Anti-tumour agents IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1990-06-20 EP disclosed