SCHEMBL9256434

SCHEMBL9256434

[CH2]C1=Cc2c(Cl)cccc21

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 3/20 0.36
CYP1A2 P05177 2/20 0.36
NPC1 O15118 1/20 0.35
TP53 P04637 1/20 0.35
HPGD P15428 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
TSHR P16473 2/20 0.35
LMNA P02545 1/20 0.35
NSD2 O96028 2/20 0.32
BCHE P06276 1/20 0.32
DAO P14920 1/20 0.32
CES1 P23141 1/20 0.32
GPR84 Q9NQS5 1/20 0.32
PTPRC P08575 1/20 0.31
ALDH1A1 P00352 3/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
NOTUM Q6P988 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31619905 0.66 ALDH1A1 (0.48) CYP1A2TP53HPGDSMN1; SMN2LMNA
SCHEMBL9682799 0.66 TSHR (0.44) CYP2A6TP53TSHRALDH1A1MEN1
SCHEMBL38867 0.64
SCHEMBL31069530 0.62 NOTUM (0.42) NPC1TP53HPGDRAB9ASMN1; SMN2
SCHEMBL440943 0.62 TSHR (0.52) CYP2A6CYP1A2TSHRLMNANOTUM
SCHEMBL29802156 0.60 CYP2A6 (0.67) CYP2A6CYP1A2NPC1TP53HPGD
SCHEMBL29883244 0.60 CYP2A6 (0.67) CYP2A6CYP1A2NPC1TP53HPGD
SCHEMBL671133 0.60 CYP2A6 (0.67) CYP2A6CYP1A2NPC1TP53HPGD
SCHEMBL9462900 0.60 CYP2A6 (0.39) CYP2A6CYP1A2NPC1TP53HPGD
SCHEMBL2095365 0.60 NOTUM (0.40) CYP2A6TSHRLMNANOTUMBLM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0490772-B1 1,4-Disubstituted piperazines, their process of preparation and pharmaceutical compositions containing them ADIR (FR) 1995-07-26 EP disclosed
EP-0490772-A1 1,4-Disubstituted piperazines, their process of preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1992-06-17 EP disclosed