SCHEMBL9256587

SCHEMBL9256587

COC(=O)C1(NC(=O)OC(C)(C)C)CCc2cc(N)ccc2C1

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GHSR Q92847 2/20 0.46
NR1H2 P55055 1/20 0.42
BACE1 P56817 3/20 0.33
PPIA P62937 2/20 0.33
HSD17B3 P37058 1/20 0.32
ESR2 Q92731 1/20 0.31
TACR1 P25103 1/20 0.31
TACR3 P29371 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
KLK5 Q9Y337 1/20 0.30
CXCR5 P32302 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9255997 0.95 GHSR (0.46) GHSRNR1H2BACE1PPIATACR1
SCHEMBL26130146 0.87 GHSR (0.47) GHSRBACE1PPIAESR2
SCHEMBL31232623 0.87 GHSR (0.47) GHSRBACE1PPIAESR2
SCHEMBL5196233 0.84 GHSR (0.61) GHSRBACE1PPIA
SCHEMBL31232553 0.83 GHSR (0.47) GHSRBACE1PPIAESR2
SCHEMBL26129956 0.83 GHSR (0.47) GHSRBACE1PPIAESR2
SCHEMBL2405143 0.82 NR1H2 (0.43) GHSRNR1H2CXCR5
SCHEMBL26401066 0.82 GHSR (0.46) GHSRBACE1PPIASMN1; SMN2
SCHEMBL26129115 0.81 GHSR (0.46) GHSRBACE1PPIASMN1; SMN2CXCR5
SCHEMBL31232508 0.81 GHSR (0.46) GHSRBACE1PPIASMN1; SMN2CXCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5378838-A FOR USE IN HUMANS MERCK & CO., INC. (US) 1995-01-03 US disclosed
WO-1994015924-A1 CHOLECYSTOKININ ANTAGONISTS MERCK & CO., INC. (US) 1994-07-21 WO disclosed