SCHEMBL9259870

SCHEMBL9259870

O=C(O)c1ncn2c1Cn1ccnc1-c1sccc1-2

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
GABRG2 P18507 15/20 0.38
GABRB3 P28472 15/20 0.38
GABRA5 P31644 14/20 0.38
AXL P30530 1/20 0.32
GABRA3 P34903 2/20 0.32
GABRA1 P14867 1/20 0.31
GABRA2 P47869 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9254656 0.85 GABRG2 (0.52) ALDH1A1CYP1A2CYP2C9CYP2C19GABRG2
SCHEMBL9660344 0.83 ALDH1A1 (0.39) ALDH1A1CYP1A2CYP2C9CYP2C19GABRG2
SCHEMBL9262794 0.81 GABRG2 (0.47) ALDH1A1CYP1A2CYP2C9CYP2C19GABRG2
SCHEMBL9661161 0.77 ALDH1A1 (0.38) ALDH1A1CYP1A2CYP2C9CYP2C19GABRG2
SCHEMBL7339291 0.76 ALDH1A1 (0.72) ALDH1A1CYP1A2CYP2C9CYP2C19GABRG2
SCHEMBL9263997 0.71 GABRG2 (0.47) ALDH1A1CYP1A2CYP2C9CYP2C19GABRG2
SCHEMBL9263686 0.69 GABRA1 (0.33) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL9259121 0.68 GABRG2 (0.68) ALDH1A1CYP1A2CYP2C9CYP2C19GABRG2
SCHEMBL15024705 0.67 ALDH1A1 (0.72) ALDH1A1CYP1A2CYP2C9CYP2C19GABRG2
SCHEMBL8871074 0.66 ALDH1A1 (0.71) ALDH1A1CYP1A2CYP2C9CYP2C19GABRG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5387585-A Treating epilepsy, anxiety, sleep disorders, schizophrnia, senile dementia HOFFMANN-LA ROCHE INC. (US) 1995-02-07 US disclosed
EP-0519307-A2 Tetracyclic Imidazodiazepines F. HOFFMANN-LA ROCHE AG (CH) 1992-12-23 EP disclosed