SCHEMBL9260283

SCHEMBL9260283

O=C(N[C@@H](CO)c1ccccc1)c1cccc2ccccc12

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 3/20 0.60
KCNA5 P22460 1/20 0.53
MMP3 P08254 1/20 0.53
HDAC8 Q9BY41 1/20 0.53
PLK1 P53350 1/20 0.51
MEN1 O00255 1/20 0.51
KMT2A Q03164 1/20 0.51
ALDH1A1 P00352 5/20 0.50
HPGD P15428 3/20 0.50
LMNA P02545 2/20 0.50
KDM4E B2RXH2 1/20 0.50
TSHR P16473 1/20 0.50
HSD17B10 Q99714 1/20 0.50
ADORA2A P29274 1/20 0.49
THRB P10828 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
MAPK13 O15264 1/20 0.49
ROCK2 O75116 1/20 0.49
RPS6KA5 O75582 1/20 0.49
MAP4K4 O95819 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22722201 0.81 HDAC8 (0.59) MMP3HDAC8PLK1MEN1KMT2A
SCHEMBL9830733 0.81 MMP3 (0.54) MMP3HDAC8PLK1MEN1KMT2A
SCHEMBL9830741 0.81 MMP3 (0.54) MMP3HDAC8PLK1MEN1KMT2A
SCHEMBL22648637 0.80 TACR3 (0.57) TACR3MEN1KMT2AALDH1A1HPGD
SCHEMBL12218397 0.79 ALDH1A1 (0.65) TACR3MMP3HDAC8PLK1ALDH1A1
SCHEMBL19813081 0.79 HPGD (0.56) TACR3KCNA5ALDH1A1HPGDLMNA
SCHEMBL5643849 0.79 NPC1 (0.55) TACR3MEN1KMT2AALDH1A1HPGD
SCHEMBL28015856 0.79 ALDH1A1 (0.60) TACR3KCNA5MEN1KMT2AALDH1A1
SCHEMBL12260876 0.78 KDM4E (0.56) TACR3KCNA5ALDH1A1HPGDLMNA
SCHEMBL8855769 0.78 KDM4E (0.51) TACR3KCNA5ALDH1A1HPGDLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995007260-A1 TETRAHYDROISOQUINOLINES AS ALPHA-2 ANTAGONISTS AND BIOGENIC AMINE UPTAKE INHIBITORS ABBOTT LABORATORIES (US) 1995-03-16 WO disclosed
US-5389638-A Nervous system disorders ABBOTT LABORATORIES (US) 1995-02-14 US disclosed