SCHEMBL9260366

SCHEMBL9260366

CCOC(=O)C(CNC(=O)C(F)(F)C(F)(F)C(=O)Nc1ccc(C(=N)N)cc1)n1ccnn1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 1/20 0.40
PDK2 Q15119 1/20 0.40
PDK3 Q15120 1/20 0.40
PDK4 Q16654 1/20 0.40
ITGB3 P05106 1/20 0.37
ITGA2B P08514 1/20 0.37
GAA P10253 2/20 0.37
KMT2A Q03164 4/20 0.36
MEN1 O00255 3/20 0.36
TSHR P16473 1/20 0.36
HTT P42858 1/20 0.36
POLB P06746 1/20 0.35
ESR2 Q92731 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
MAPT P10636 3/20 0.35
RGS12 O14924 1/20 0.35
ALDH1A1 P00352 1/20 0.35
F10 P00742 2/20 0.35
F2 P00734 2/20 0.35
PRSS1 P07477 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6979019 0.74 ITGB3 (0.39) ITGB3ITGA2BGAATSHRHTT
SCHEMBL6982396 0.74 ITGB3 (0.35) ITGB3ITGA2BGAATSHRALDH1A1
SCHEMBL9558850 0.68 ITGB3 (0.53) ITGB3ITGA2BF10F2PRSS1
SCHEMBL9263893 0.68 KLK1 (0.38) ITGB3ITGA2BF2PRSS1PRSS2
SCHEMBL4414766 0.64 F7 (0.57) ITGB3ITGA2BF10F2PRSS1
SCHEMBL7348941 0.64 ITGB3 (0.57) ITGB3ITGA2BGAAMAPT
SCHEMBL7347870 0.64 ITGB3 (0.57) ITGB3ITGA2BGAAHTTMAPT
SCHEMBL6981952 0.63 ALDH1A1 (0.49) ITGB3ITGA2BKMT2AHTTMAPT
SCHEMBL6978796 0.62 ITGB3 (0.48) ITGB3ITGA2BGAATSHRPOLB
SCHEMBL1542395 0.62 PDK1 (0.74) PDK1PDK2PDK3PDK4GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5378727-A ADMINISTERING TO MAMMALS G. D. SEARLE & CO. (US) 1995-01-03 US disclosed
US-5254573-A Substituted heterocyclic derivatives useful as platelet aggregation inhibitors MONSANTO COMPANY (US) 1993-10-19 US disclosed
EP-0539343-A1 Substituted heterocyclic derivatives useful as platelet aggregation inhibitors MONSANTO COMPANY (US) 1993-04-28 EP disclosed