SCHEMBL9260520

SCHEMBL9260520

O=c1cc(-c2ccccc2)sn1-c1ccc(N(C(F)(F)F)S(=O)(=O)C(F)(F)F)cc1

nearest known ligand 0.33

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NR1H3 Q13133 2/20 0.33
NR1H2 P55055 1/20 0.33
PMM2 O15305 1/20 0.32
MPI P34949 1/20 0.32
PHOSPHO1 Q8TCT1 1/20 0.32
PTGS2 P35354 1/20 0.31
G6PD P11413 1/20 0.30
TLR9 Q9NR96 1/20 0.30
KAT2B Q92831 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9263852 0.72 PHOSPHO1 (0.47) PMM2MPIPHOSPHO1G6PDKAT2B
SCHEMBL176126 0.72 NR1H3 (0.45) NR1H3NR1H2PTGS2
SCHEMBL9256001 0.71 KDM4E (0.40) KAT2B
SCHEMBL9262493 0.69 MAPT (0.46) PMM2MPIPHOSPHO1
SCHEMBL9258084 0.66 ALDH1A1 (0.43) G6PDTLR9KAT2B
SCHEMBL9256085 0.64 PMM2 (0.45) PMM2MPIPHOSPHO1KAT2B
SCHEMBL9263510 0.64 SMN1; SMN2 (0.60) MPIPHOSPHO1KAT2B
SCHEMBL8818175 0.63 CA2 (0.40) NR1H3NR1H2PTGS2
SCHEMBL9265563 0.60 KDM4E (0.40)
SCHEMBL8080054 0.59 HSD17B10 (0.41) G6PD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5411977-A Substituted 2,5-diaryl-4-isothiazolin-3-ones as antiinflammatory and antithrombotic agents THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1995-05-02 US disclosed