SCHEMBL176126

SCHEMBL176126

O=S(=O)(N(c1ccccc1)C(F)(F)F)C(F)(F)F

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H3 Q13133 4/20 0.45
NR1H2 P55055 2/20 0.45
ALDH1A1 P00352 2/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
CA2 P00918 2/20 0.36
CA9 Q16790 2/20 0.36
CA1 P00915 1/20 0.36
CA5A P35218 1/20 0.36
RORC P51449 3/20 0.35
APOBEC3G Q9HC16 1/20 0.34
PKM P14618 1/20 0.34
NR1I2 O75469 5/20 0.34
PTGS1 P23219 1/20 0.34
PTGS2 P35354 1/20 0.34
RORA P35398 2/20 0.33
RORB Q92753 2/20 0.33
NR1H4 Q96RI1 2/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8818175 0.80 CA2 (0.40) NR1H3NR1H2CA2CA9CA1
SCHEMBL28103135 0.80 NR1H3 (0.43) NR1H3NR1H2ALDH1A1MEN1KMT2A
SCHEMBL10622844 0.79 NR1H3 (0.45) NR1H3NR1H2ALDH1A1MEN1KMT2A
SCHEMBL27609289 0.79 CA2 (0.45) NR1H3NR1H2ALDH1A1MEN1KMT2A
SCHEMBL4306577 0.79 NR1H3 (0.49) NR1H3NR1H2ALDH1A1MEN1KMT2A
SCHEMBL64494 0.78 CA2 (0.43) NR1H3ALDH1A1MEN1KMT2ACA2
SCHEMBL13096335 0.78 PKM (0.45) NR1H3ALDH1A1MEN1KMT2ACA2
SCHEMBL6917666 0.78 NR1H3 (0.69) NR1H3NR1H2ALDH1A1RORCAPOBEC3G
SCHEMBL15082546 0.75 ALDH1A1 (0.37) NR1H3ALDH1A1MEN1KMT2ACA2
SCHEMBL14331424 0.75 HSP90AA1 (0.48) NR1H3NR1H2ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 121 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4735431-A2 MK2 INHIBITORS AND METHODS OF MAKING AND USING THE SAME GILEAD SCIENCES, INC. (US) 2026-05-06 EP disclosed
EP-4695260-A1 KRAS MODULATING COMPOUNDS GILEAD SCIENCES, INC. (US) 2026-02-18 EP disclosed
US-20250388585-A1 PRMT5 INHIBITORS AND USES THEREOF GILEAD SCIENCES INC (US) 2025-12-25 US disclosed
US-12448388-B2 PRMT5 inhibitors and uses thereof GILEAD SCIENCES, INC. (US) 2025-10-21 US disclosed
US-20250230168-A1 AZASPIRO WRN INHIBITORS GILEAD SCIENCES, INC. 2025-07-17 US disclosed
WO-2025137640-A1 AZASPIRO WRN INHIBITORS GILEAD SCIENCES, INC. (US) 2025-06-26 WO disclosed
US-20250154172-A1 PRMT5 INHIBITORS AND USES THEREOF GILEAD SCIENCES, INC. 2025-05-15 US disclosed
US-20250092017-A1 2-PIPERIDYL OR 2-PYRAZOLYL SUBSTITUTED PYRIMIDINE COMPOUND SERVING AS EGFR INHIBITOR Suzhou Puhe BioPharma Co., Ltd. (CN) 2025-03-20 US disclosed
US-20250051309-A1 MK2 INHIBITORS AND METHODS OF MAKING AND USING THE SAME GILEAD SCIENCES, INC. 2025-02-13 US disclosed
WO-2025006568-A2 MK2 INHIBITORS AND METHODS OF MAKING AND USING THE SAME GILEAD SCIENCES, INC. (US) 2025-01-02 WO disclosed
WO-2010071885-A1 PYRROLOTRIAZINES AS ALK AND JAK2 INHIBITORS CEPHALON, INC. (US) 2010-06-24 WO disclosed
US-20100093694-A1 Compounds for the Treatment of Hepatitis C BRISTOL-MYERS SQUIBB COMPANY 2010-04-15 US disclosed
WO-2010030592-A1 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C BRISTOL-MYERS SQUIBB COMPANY (US) 2010-03-18 WO disclosed
WO-2010030538-A2 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C BRISTOL-MYERS SQUIBB COMPANY (US) 2010-03-18 WO disclosed
US-20100063068-A1 Compounds for the Treatment of Hepatitis C BRISTOL-MYERS SQUIBB COMPANY 2010-03-11 US disclosed
US-20080312286-A1 Indanone Potentiators of Metabotropic Glutamate Receptors MERCK SHARP & DOHME CORP. 2008-12-18 US disclosed
US-20070149577-A1 Compounds with medicinal effects due to interaction with the glucocorticoid receptor N.V. ORGANON (NL) 2007-06-28 US disclosed
US-20040122001-A1 Pharmaceutical compounds ELI LILLY AND COMPANY 2004-06-24 US disclosed
EP-1345930-A2 PHARMACEUTICAL COMPOUNDS ELI LILLY AND COMPANY (US) 2003-09-24 EP disclosed
WO-2002050067-A2 PHARMACEUTICAL HETEROCYCLIC COMPOUNDS ELI LILLY AND COMPANY (US) 2002-06-27 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (11 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250388585-A1 PRMT5 INHIBITORS AND USES THEREOF PRMT1, PRMT5, PRMT6 NR1H3 2328/4885NR1H2 2419/4885ALDH1A1 3522/4885
US-20250230168-A1 AZASPIRO WRN INHIBITORS WRN, RECQL, BLM NR1H3 3424/4885NR1H2 2809/4885ALDH1A1 1316/4885
US-20070149577-A1 Compounds with medicinal effects due to interaction with the glucocorticoid receptor NR3C1, NR3C2, MC2R NR1H3 90/4885NR1H2 97/4885ALDH1A1 1050/4885
US-20250092017-A1 2-PIPERIDYL OR 2-PYRAZOLYL SUBSTITUTED PYRIMIDINE COMPOUND SERVING AS EGFR INHIBITOR EGFR, ERBB2, ERBB4 NR1H3 3657/4885NR1H2 3263/4885ALDH1A1 3675/4885
US-20080312286-A1 Indanone Potentiators of Metabotropic Glutamate Receptors GRM2, GRIK2, GRM1 NR1H3 232/4885NR1H2 173/4885ALDH1A1 2475/4885
US-20250154172-A1 PRMT5 INHIBITORS AND USES THEREOF PRMT5, PRMT1, PRMT9 NR1H3 3830/4885NR1H2 3688/4885ALDH1A1 3108/4885
US-20100063068-A1 Compounds for the Treatment of Hepatitis C HAVCR2, HCCS, SLC10A1 NR1H3 43/4885NR1H2 88/4885ALDH1A1 447/4885
US-12448388-B2 PRMT5 inhibitors and uses thereof PRMT5, PRMT1, PRMT9 NR1H3 3875/4885NR1H2 3775/4885ALDH1A1 3212/4885
US-20250051309-A1 MK2 INHIBITORS AND METHODS OF MAKING AND USING THE SAME DUSP2, MKNK2, DUSP22 NR1H3 1729/4885NR1H2 1042/4885ALDH1A1 4336/4885
US-20100093694-A1 Compounds for the Treatment of Hepatitis C HAVCR2, HCCS, SLC10A1 NR1H3 56/4885NR1H2 83/4885ALDH1A1 239/4885
US-20040122001-A1 Pharmaceutical compounds CYP2D6, LPXN, CYP1B1 NR1H3 821/4885NR1H2 783/4885ALDH1A1 1563/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.