SCHEMBL9260683

SCHEMBL9260683

O=C1Cn2ccnc2-c2c(Br)cccc2N1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.34
TSHR P16473 1/20 0.34
TGM2 P21980 1/20 0.34
KDR P35968 3/20 0.33
CDK5 Q00535 2/20 0.32
CDK5R1 Q15078 2/20 0.32
AHR P35869 1/20 0.32
PDK2 Q15119 1/20 0.32
MAPK1 P28482 1/20 0.32
LMNA P02545 1/20 0.32
GAA P10253 1/20 0.32
CCNB2 O95067 1/20 0.32
CDK1 P06493 1/20 0.32
CCNB1 P14635 1/20 0.32
GSK3B P49841 1/20 0.32
CCNB3 Q8WWL7 1/20 0.32
HRH1 P35367 2/20 0.31
RET P07949 1/20 0.31
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9260664 0.85 GRIA1 (0.42) ALDH1A1TSHRKDRLMNAHRH1
SCHEMBL9261989 0.84 CES1 (0.42) ALDH1A1TSHRTGM2CDK5CDK5R1
SCHEMBL9267469 0.79
SCHEMBL9267374 0.77 KDR (0.46) ALDH1A1TSHRKDRCDK5CDK5R1
SCHEMBL9715259 0.70 KMT2A (0.52) ALDH1A1CDK5CDK5R1LMNACCNB2
SCHEMBL9259415 0.68 GABRA1 (0.40) CDK5CDK5R1GSK3BADRA1A
SCHEMBL5739203 0.66 BRD4 (0.45) KDRCDK5CDK5R1AHRPDK2
Hydrochloric Acid SCHEMBL10369856 0.65 BRD4 (0.44) KDRCDK5CDK5R1AHRPDK2
SCHEMBL9050196 0.64 MMP12 (0.39) ALDH1A1CDK5CDK5R1AHRPDK2
SCHEMBL5024271 0.64

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5387585-A Treating epilepsy, anxiety, sleep disorders, schizophrnia, senile dementia HOFFMANN-LA ROCHE INC. (US) 1995-02-07 US disclosed
EP-0519307-A2 Tetracyclic Imidazodiazepines F. HOFFMANN-LA ROCHE AG (CH) 1992-12-23 EP disclosed