SCHEMBL9263233

SCHEMBL9263233

COc1ccccc1-n1c(=O)ccc2ccccc21

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 1/20 0.51
MGLL Q99685 1/20 0.47
CA12 O43570 1/20 0.47
BRD4 O60885 1/20 0.47
BRPF1 P55201 1/20 0.47
CA9 Q16790 1/20 0.47
KAT2B Q92831 1/20 0.47
BRD9 Q9H8M2 1/20 0.47
TSHR P16473 1/20 0.47
ALDH1A1 P00352 2/20 0.47
KMT2A Q03164 2/20 0.47
KDM4E B2RXH2 1/20 0.47
MAPT P10636 1/20 0.47
HPGD P15428 1/20 0.47
HTT P42858 1/20 0.47
MEN1 O00255 1/20 0.47
APLNR P35414 4/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
METAP2 P50579 1/20 0.43
PTGS2 P35354 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17505155 0.75 CA12 (0.47) CA12BRD4BRPF1CA9KAT2B
SCHEMBL9270290 0.75 POLB (0.50) CA12BRD4BRPF1CA9KAT2B
SCHEMBL29009659 0.75 CA12 (0.47) SCN9AMGLLCA12BRD4BRPF1
SCHEMBL23075577 0.74 DRD2 (0.42) MGLLTSHRALDH1A1KMT2AKDM4E
SCHEMBL11693860 0.74 LMNA (0.53) MGLLCA12BRD4BRPF1CA9
SCHEMBL23075579 0.73 ALDH1A1 (0.59) TSHRALDH1A1KMT2AKDM4EHPGD
SCHEMBL5150754 0.72 KMT2A (0.59) MGLLCA12BRD4BRPF1CA9
SCHEMBL30440787 0.72 ALDH1A1 (0.49) CA12BRD4BRPF1CA9KAT2B
SCHEMBL28181208 0.72 MGLL (0.47) MGLLCA12CA9ALDH1A1KMT2A
SCHEMBL16296570 0.71 SCN9A (0.61) SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995003300-A1 HETEROARYL QUINOLINES AS INHIBITORS OF LEUKOTRIENE BIOSYNTHESIS MERCK FROSST CANADA INC. (CA) 1995-02-02 WO disclosed