SCHEMBL9267705

SCHEMBL9267705

C=CCc1oc2ccccc2c1C(=O)c1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EYA3 Q99504 8/20 0.55
SLC22A12 Q96S37 2/20 0.55
CYP2C19 P33261 7/20 0.51
PTPN1 P18031 2/20 0.50
CYP2C9 P11712 5/20 0.48
KMT2A Q03164 3/20 0.48
TTR P02766 3/20 0.48
MEN1 O00255 2/20 0.48
ABCB11 O95342 2/20 0.48
LMNA P02545 2/20 0.48
PGR P06401 2/20 0.48
ADRA2A P08913 2/20 0.48
TBXA2R P21731 2/20 0.48
OPRM1 P35372 2/20 0.48
SLC6A3 Q01959 2/20 0.48
BIRC5 O15392 1/20 0.48
HTR1A P08908 1/20 0.48
DRD1 P21728 1/20 0.48
PTGS1 P23219 1/20 0.48
SLC6A2 P23975 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2141567 0.90 EYA3 (0.69) EYA3SLC22A12CYP2C19PTPN1CYP2C9
SCHEMBL4430343 0.89 EYA3 (0.44) EYA3SLC22A12CYP2C19PTPN1CYP2C9
SCHEMBL10599107 0.86 CYP2C19 (0.63) EYA3SLC22A12CYP2C19PTPN1CYP2C9
SCHEMBL10598815 0.84 EYA3 (0.54) EYA3SLC22A12CYP2C19PTPN1CYP2C9
SCHEMBL9605230 0.84 EYA3 (0.43) EYA3SLC22A12CYP2C19PTPN1CYP2C9
SCHEMBL9287304 0.80 EYA3 (0.53) EYA3SLC22A12CYP2C19PTPN1CYP2C9
SCHEMBL1287913 0.80 EYA3 (0.81) EYA3SLC22A12CYP2C19PTPN1CYP2C9
SCHEMBL10602010 0.79 CYP2C19 (0.46) EYA3SLC22A12CYP2C19PTPN1CYP2C9
SCHEMBL11734971 0.79 EYA3 (0.57) EYA3SLC22A12CYP2C19PTPN1CYP2C9
SCHEMBL9284220 0.78 MAPT (0.56) PTPN1KMT2AMAPTALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0448850-B1 2-Alkyl-3-benzoylbenzofurans useful for treating cardiac arrhythmia TARO PHARMA IND (IL) 1995-08-30 EP claimed
EP-0338746-B1 2-Alkyl-3-benzoylbenzofurans and pharmaceutical compositions containing them TARO PHARMA IND (IL) 1994-08-31 EP claimed
EP-0448850-A1 2-Alkyl-3-benzoylbenzofurans useful for treating cardiac arrhythmia Taro Pharmaceutical Industries Ltd. (IL) 1991-10-02 EP claimed
US-4975458-A 2-alkyl-3-benzoylbenzofurans useful for treating cardiac arrhythmia TARO PHARMACEUTICALS INDUSTRIES, LTD. (IL) 1990-12-04 US claimed
EP-0338746-A1 2-Alkyl-3-benzoylbenzofurans and pharmaceutical compositions containing them Taro Pharmaceutical Industries Ltd. (IL) 1989-10-25 EP claimed
US-4831054-A 2-Alkyl-3-benzoylbenzofurans useful for treating cardiac arrhythmia TARO PHARMACEUTICALS, LTD. (IL) 1989-05-16 US claimed
EP-0448850-B1 2-Alkyl-3-benzoylbenzofurans useful for treating cardiac arrhythmia TARO PHARMA IND (IL) 1995-08-30 EP disclosed
EP-0448850-B1 2-Alkyl-3-benzoylbenzofurans useful for treating cardiac arrhythmia TARO PHARMA IND (IL) 1995-08-30 EP disclosed
EP-0338746-B1 2-Alkyl-3-benzoylbenzofurans and pharmaceutical compositions containing them TARO PHARMA IND (IL) 1994-08-31 EP disclosed
EP-0338746-B1 2-Alkyl-3-benzoylbenzofurans and pharmaceutical compositions containing them TARO PHARMA IND (IL) 1994-08-31 EP disclosed
EP-0448850-A1 2-Alkyl-3-benzoylbenzofurans useful for treating cardiac arrhythmia Taro Pharmaceutical Industries Ltd. (IL) 1991-10-02 EP disclosed
EP-0448850-A1 2-Alkyl-3-benzoylbenzofurans useful for treating cardiac arrhythmia Taro Pharmaceutical Industries Ltd. (IL) 1991-10-02 EP disclosed
US-4975458-A 2-alkyl-3-benzoylbenzofurans useful for treating cardiac arrhythmia TARO PHARMACEUTICALS INDUSTRIES, LTD. (IL) 1990-12-04 US disclosed
US-4975458-A 2-alkyl-3-benzoylbenzofurans useful for treating cardiac arrhythmia TARO PHARMACEUTICALS INDUSTRIES, LTD. (IL) 1990-12-04 US disclosed
EP-0338746-A1 2-Alkyl-3-benzoylbenzofurans and pharmaceutical compositions containing them Taro Pharmaceutical Industries Ltd. (IL) 1989-10-25 EP disclosed
EP-0338746-A1 2-Alkyl-3-benzoylbenzofurans and pharmaceutical compositions containing them Taro Pharmaceutical Industries Ltd. (IL) 1989-10-25 EP disclosed
US-4831054-A 2-Alkyl-3-benzoylbenzofurans useful for treating cardiac arrhythmia TARO PHARMACEUTICALS, LTD. (IL) 1989-05-16 US disclosed
US-4831054-A 2-Alkyl-3-benzoylbenzofurans useful for treating cardiac arrhythmia TARO PHARMACEUTICALS, LTD. (IL) 1989-05-16 US disclosed