SCHEMBL9280946

SCHEMBL9280946

NCC(O)(Oc1cccc(C(F)(F)F)c1)c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAOB P27338 2/20 0.48
AOC3 Q16853 1/20 0.48
KIF11 P52732 2/20 0.47
PPARG P37231 2/20 0.47
PPARA Q07869 1/20 0.47
KDM4E B2RXH2 2/20 0.46
MRGPRX4 Q96LA9 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
PNMT P11086 1/20 0.42
TAAR1 Q96RJ0 1/20 0.41
ALDH1A1 P00352 1/20 0.41
IDO1 P14902 2/20 0.41
ADORA2A P29274 1/20 0.40
TDO2 P48775 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11527555 0.73 KIF11 (0.51) MAOBAOC3KIF11PPARGPPARA
SCHEMBL23519064 0.71 PPARG (0.51) PPARGPPARAKDM4EMRGPRX4ALDH1A1
SCHEMBL9546526 0.71 L3MBTL1 (0.55) MAOBKIF11PPARGPPARAL3MBTL1
SCHEMBL7797664 0.70 KIF11 (0.41) KIF11TAAR1
SCHEMBL4008943 0.70 PPARG (0.52) PPARGPPARAKDM4EMRGPRX4ALDH1A1
SCHEMBL10599070 0.70 TSHR (0.45) MAOBAOC3PPARGPPARAKDM4E
SCHEMBL2737127 0.70 L3MBTL1 (0.47) MAOBAOC3PPARGPPARAKDM4E
SCHEMBL3524104 0.69 L3MBTL1 (0.59) MAOBAOC3KDM4EMRGPRX4L3MBTL1
SCHEMBL3054166 0.69 TAAR1 (0.45) KIF11KDM4ETAAR1ALDH1A1
SCHEMBL4214531 0.69 TSHR (0.54) MAOBAOC3PPARGPPARAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5514694-A ENZYME INHIBITORS GEORGIA TECH RESEARCH CORP (US) 1996-05-07 US disclosed
EP-0650368-A1 USE OF CALPAIN INHIBITORS IN THE INHIBITION AND TREATMENT OF MEDICAL CONDITIONS ASSOCIATED WITH INCREASED CALPAIN ACTIVITY CORTEX PHARMACEUTICALS, INC. (US) 1995-05-03 EP disclosed
WO-1994000095-A2 USE OF CALPAIN INHIBITORS IN THE INHIBITION AND TREATMENT OF MEDICAL CONDITIONS ASSOCIATED WITH INCREASED CALPAIN ACTIVITY CORTEX PHARMACEUTICALS, INC. (US) 1994-01-06 WO disclosed