SCHEMBL9288758

SCHEMBL9288758

Cc1cccc(N(C(N)=O)[C@H]2N=C(NCCN(C)C)c3ccccc3N(C)C2=O)c1

nearest known ligand 0.39

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 17/20 0.39
KCNH2 Q12809 1/20 0.38
NOTCH1 P46531 1/20 0.36
NOTCH3 Q9UM47 1/20 0.36
SYK P43405 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8863378 0.79 CCKBR (0.55) CCKBRKCNH2NOTCH1NOTCH3
SCHEMBL7626581 0.79 CCKBR (0.55) CCKBRKCNH2NOTCH1NOTCH3
SCHEMBL7819355 0.78 CCKBR (0.65) CCKBRKCNH2
Hydrochloric Acid SCHEMBL7824167 0.77 CCKBR (0.64) CCKBRKCNH2
SCHEMBL7312531 0.77 CCKBR (0.40) CCKBRKCNH2NOTCH1NOTCH3
SCHEMBL9368599 0.76 CCKBR (0.57) CCKBRKCNH2
SCHEMBL7827288 0.76 CCKBR (0.58) CCKBRKCNH2
SCHEMBL7308632 0.75 CCKBR (0.41) CCKBRKCNH2NOTCH1NOTCH3
Hydrochloric Acid SCHEMBL9385743 0.73 CCKBR (0.49) CCKBRKCNH2
SCHEMBL9272997 0.68 CCKBR (0.40) CCKBR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0652871-A1 BENZODIAZEPINE DERIVATIVES MERCK SHARP & DOHME LTD. (GB) 1995-05-17 EP claimed