SCHEMBL9296383

SCHEMBL9296383

O=C1CCSCC1Cc1ccccc1Br

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP27A1 Q02318 1/20 0.43
CYP24A1 Q07973 1/20 0.43
PTGS1 P23219 1/20 0.36
PTGS2 P35354 1/20 0.36
DRD2 P14416 1/20 0.35
DRD3 P35462 1/20 0.35
TAAR1 Q96RJ0 1/20 0.33
GSK3B P49841 1/20 0.32
ATM Q13315 1/20 0.32
IDO1 P14902 2/20 0.32
P2RX7 Q99572 1/20 0.32
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
CA4 P22748 1/20 0.31
CA6 P23280 1/20 0.31
MMP1 P03956 1/20 0.31
MMP2 P08253 1/20 0.31
MMP9 P14780 1/20 0.31
MMP12 P39900 1/20 0.31
KDM1A O60341 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29169537 0.76 PTGS1 (0.52) CYP27A1CYP24A1PTGS1PTGS2ATM
SCHEMBL30825588 0.76 PTGS1 (0.52) CYP27A1CYP24A1PTGS1PTGS2ATM
SCHEMBL9296486 0.76 PTGS1 (0.52) CYP27A1CYP24A1PTGS1PTGS2ATM
SCHEMBL2488144 0.75 PTGS1 (0.51) CYP27A1CYP24A1PTGS1PTGS2CA1
SCHEMBL9296275 0.74 PTGS1 (0.50) CYP27A1CYP24A1PTGS1PTGS2CA1
SCHEMBL13867248 0.72 PTGS2 (0.37) PTGS1PTGS2
Hydrochloric Acid SCHEMBL9296314 0.72 CYP27A1 (0.40) CYP27A1CYP24A1PTGS1PTGS2DRD2
SCHEMBL30569684 0.68 CYP27A1 (0.41) CYP27A1CYP24A1TAAR1ATMIDO1
SCHEMBL7089627 0.68 CYP27A1 (0.37) CYP27A1CYP24A1PTGS1PTGS2DRD2
SCHEMBL9296600 0.67 TACR1 (0.52) ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5276053-A Dibenzothiopyranylamines WARNER-LAMBERT COMPANY (US) 1994-01-04 US disclosed
US-5180736-A Treatment and prevention of brain disorders WARNER-LAMBERT COMPANY (US) 1993-01-19 US disclosed
US-5071853-A Amine-substituted hexahydroindeno(2,1-b)pyrroles, -indeno(2,1-c)pyridines or -indeno(2,1-d)azepines; cerebral ischemia or infarction WARNER-LAMBERT COMPANY 1991-12-10 US disclosed
EP-0388977-A2 Polycyclic amines useful as cerebrovascular agents WARNER-LAMBERT COMPANY (US) 1990-09-26 EP disclosed