SCHEMBL9300367

SCHEMBL9300367

Cc1cc(S)nc2ccnn12

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 3/20 0.43
KCNN3 Q9UGI6 4/20 0.35
CCNT1 O60563 8/20 0.33
CDK9 P50750 8/20 0.33
KCNN1 Q92952 1/20 0.33
KCNN2 Q9H2S1 1/20 0.33
CDK7 P50613 3/20 0.32
CCNH P51946 3/20 0.32
CDK4 P11802 2/20 0.32
CCND1 P24385 2/20 0.32
PIK3CG P48736 1/20 0.32
ALDH1A1 P00352 1/20 0.32
CBLB Q13191 1/20 0.31
HTR2C P28335 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3460690 0.80 PIK3CG (0.48) PDE10APIK3CGALDH1A1
SCHEMBL29344715 0.77 PDE10A (0.67) PDE10AKCNN3CCNT1CDK9KCNN1
SCHEMBL20664459 0.77 PDE10A (0.43) PDE10AKCNN3CCNT1CDK9KCNN1
SCHEMBL13073900 0.77 PDE10A (0.43) PDE10AKCNN3CCNT1CDK9KCNN1
SCHEMBL12364000 0.77 PDE10A (0.43) PDE10AKCNN3CCNT1CDK9KCNN1
SCHEMBL25807858 0.74 CCNT1 (0.54) CCNT1CDK9CDK7CCNHCDK4
SCHEMBL21849086 0.74 KDM4E (0.42) PDE10AKCNN3CCNT1CDK9KCNN1
SCHEMBL17690933 0.74 PRKAB2 (0.49) PDE10AKCNN3CCNT1CDK9KCNN1
SCHEMBL9301157 0.73 PDE10A (0.43) PDE10AKCNN3CCNT1CDK9PIK3CG
SCHEMBL21212195 0.73 PDE10A (0.51) PDE10ACCNT1CDK9CDK7CCNH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5319140-A Antibiotics HOFFMANN-LA ROCHE INC. (US) 1994-06-07 US disclosed
US-5138066-A Intermediates for cephalosporins with sulfur-containing oxyimino side chain HOFFMANN-LA ROCHE, INC. (US) 1992-08-11 US disclosed
US-5073550-A Bactericides HOFFMANN-LA ROCHE INC. (US) 1991-12-17 US disclosed
US-5036064-A Antibiotics HOFFMANN-LA ROCHE INC. (US) 1991-07-30 US disclosed
EP-0303172-A2 Oxyimino-cephalosporins F. HOFFMANN-LA ROCHE AG (CH) 1989-02-15 EP disclosed