SCHEMBL9300629

SCHEMBL9300629

CCOC(=O)C1CC(=O)c2ccc(OC)cc2C1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.69
KMT2A Q03164 4/20 0.69
KDM4E B2RXH2 3/20 0.69
HTR2A P28223 3/20 0.48
HTR2C P28335 3/20 0.48
DRD2 P14416 2/20 0.48
MEN1 O00255 3/20 0.47
MAPT P10636 2/20 0.47
GAA P10253 2/20 0.47
HPGD P15428 1/20 0.47
HSD17B10 Q99714 1/20 0.47
POLB P06746 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
PPARG P37231 3/20 0.46
METAP1 P53582 2/20 0.45
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
TSHR P16473 2/20 0.43
MAPK1 P28482 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9370726 0.85 ALDH1A1 (0.54) ALDH1A1KMT2AKDM4EMEN1MAPT
SCHEMBL15774873 0.84 KMT2A (0.64) ALDH1A1KMT2AKDM4EMEN1MAPT
SCHEMBL15774975 0.83 ALDH1A1 (0.55) ALDH1A1KMT2AKDM4EHTR2AHTR2C
SCHEMBL344573 0.82 CYP19A1 (0.50) ALDH1A1KMT2AKDM4EHTR2AHTR2C
SCHEMBL344572 0.82 CYP19A1 (0.50) ALDH1A1KMT2AKDM4EHTR2AHTR2C
SCHEMBL4730776 0.81 ALDH1A1 (0.70) ALDH1A1KMT2AKDM4EMEN1MAPT
SCHEMBL9344657 0.80 ALDH1A1 (0.61) ALDH1A1KMT2AKDM4EMEN1MAPT
SCHEMBL630214 0.78 DRD2 (0.51) ALDH1A1KMT2AKDM4EDRD2MEN1
SCHEMBL9688032 0.78 MTNR1A (0.54) ALDH1A1KMT2AKDM4EDRD2MEN1
SCHEMBL7289390 0.78 DRD2 (0.51) ALDH1A1KMT2AKDM4EDRD2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014086697-A1 SUBSTITUTED THIAZOLE COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2014-06-12 WO disclosed
US-5308852-A Cardiovascular disorders MERCK FROSST CANADA, INC. (CA) 1994-05-03 US disclosed
EP-0579304-A1 Heteroarylnaphthalenes as inhibitors of leukotriene biosynthesis MERCK FROSST CANADA INC. (CA) 1994-01-19 EP disclosed
WO-1994000444-A1 HETEROARYLNAPHTHALENES AS INHIBITORS OF LEUKOTRIENE BIOSYNTHESIS MERCK FROSST CANADA INC. (CA) 1994-01-06 WO disclosed