SCHEMBL9301158

SCHEMBL9301158

OC(COc1ccc(F)cc1)CN1CCN(CCCC(c2ccc(C(F)(F)F)cc2)c2ccc(C(F)(F)F)cc2)CC1

nearest known ligand 0.67

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CACNA1G O43497 7/20 0.67
CYP2D6 P10635 4/20 0.60
KCNH2 Q12809 5/20 0.54
MAPT P10636 1/20 0.53
TSHR P16473 1/20 0.51
SCN1A P35498 2/20 0.50
SCN5A Q14524 2/20 0.50
SCN9A Q15858 2/20 0.50
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
KDM4E B2RXH2 1/20 0.49
GLA P06280 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9187274 0.93 MAPT (0.60) CACNA1GKCNH2MAPTTSHRMEN1
SCHEMBL9301397 0.89 MAPT (0.57) CACNA1GCYP2D6KCNH2MAPTTSHR
SCHEMBL9301814 0.88 CYP2D6 (0.54) CACNA1GCYP2D6KCNH2MAPTSCN1A
SCHEMBL9193205 0.88 L3MBTL1 (0.59) CACNA1GCYP2D6KCNH2MAPTTSHR
SCHEMBL10379764 0.88 L3MBTL1 (0.62) CACNA1GCYP2D6KCNH2MAPTTSHR
SCHEMBL9301602 0.88 TSHR (0.64) CACNA1GCYP2D6KCNH2MAPTTSHR
SCHEMBL9300891 0.88 TSHR (0.64) CACNA1GCYP2D6KCNH2MAPTTSHR
SCHEMBL9271436 0.88 CACNA1G (0.67) CACNA1GKCNH2MAPTTSHRMEN1
SCHEMBL9301487 0.87 CYP2D6 (0.55) CACNA1GCYP2D6KCNH2MAPTSCN1A
SCHEMBL9301847 0.86 CACNA1G (0.64) CACNA1GCYP2D6KCNH2SCN1ASCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5342839-A Useful for therapy of oxygen deficiency diseases of the brain BASF AKTIENGESELLSCHAFT (DE) 1994-08-30 US disclosed
WO-1990003371-A1 2-HYDROXY-3-PHENOXY-PROPYL-SUBSTITUTED PIPERAZINES AND HOMOPIPERAZINES, THEIR MANUFACTURE AND USE BASF AKTIENGESELLSCHAFT (DE) 1990-04-05 WO disclosed