SCHEMBL9301414

SCHEMBL9301414

O=S(=O)(NNc1cccc(Cl)c1)c1ccc(CBr)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 9/20 0.48
CYP19A1 P11511 2/20 0.48
ALOX15 P16050 1/20 0.46
ALDH1A1 P00352 3/20 0.43
GFER P55789 2/20 0.43
KDM4E B2RXH2 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
GAA P10253 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
HPGD P15428 1/20 0.43
ALOX12 P18054 1/20 0.43
CYP2C19 P33261 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
APOBEC3G Q9HC16 1/20 0.43
PGR P06401 2/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
LIMK2 P53671 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9305039 0.86 CYP19A1 (0.67) CYP19A1ALOX15ALDH1A1CYP1A2CYP3A4
SCHEMBL27492176 0.82 PGR (0.61) IDO1CYP19A1ALDH1A1GFERKDM4E
SCHEMBL28692275 0.69 KMT2A (0.67) ALDH1A1GAAMEN1KMT2APKM
SCHEMBL8795345 0.67 MAPT (0.61) IDO1ALOX15ALDH1A1GFERCYP3A4
SCHEMBL2251010 0.67 KAT6A (0.59) IDO1CYP19A1ALDH1A1GFERKDM4E
SCHEMBL9301411 0.67 NPC1 (0.50) HPGDMEN1KMT2A
SCHEMBL27599728 0.67 PNMT (0.50) IDO1CYP3A4
SCHEMBL3791521 0.66 PGR (0.81) CYP19A1ALOX15ALDH1A1CYP1A2CYP3A4
SCHEMBL343776 0.66 HTR6 (0.73) CYP19A1ALOX15ALDH1A1CYP1A2CYP3A4
SCHEMBL14937571 0.66 PGR (0.72) CYP19A1ALOX15ALDH1A1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5314880-A Platelet activating factor antagonist BRITISH BIO-TECHNOLOGY LIMITED (GB) 1994-05-24 US disclosed
EP-0468971-A1 NOVEL BENZIMIDAZOLE DERIVATIVES BRITISH BIO-TECHNOLOGY LIMITED (GB) 1992-02-05 EP disclosed
WO-1990009997-A1 NOVEL BENZIMIDAZOLE DERIVATIVES BRITISH BIO-TECHNOLOGY LIMITED (GB) 1990-09-07 WO disclosed