SCHEMBL9301411

SCHEMBL9301411

NS(=O)(=O)c1ccc(CBr)cc1Nc1cccc(Cl)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.50
HPGD P15428 1/20 0.50
HTT P42858 1/20 0.50
PTGES2 Q9H7Z7 4/20 0.41
P2RY2 P41231 1/20 0.41
P2RY4 P51582 1/20 0.41
P2RY12 Q9H244 1/20 0.41
CA9 Q16790 3/20 0.40
CA1 P00915 3/20 0.40
CA2 P00918 3/20 0.40
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
CA12 O43570 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
PTGS1 P23219 2/20 0.40
PTGS2 P35354 2/20 0.40
MT-CO2 P00403 1/20 0.40
FADS1 O60427 1/20 0.40
MAPT P10636 1/20 0.38
P2RX4 Q99571 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24051716 0.71 CA1 (0.44) PTGES2CA9CA1CA2CA12
SCHEMBL9305039 0.69 CYP19A1 (0.67) MEN1KMT2A
SCHEMBL7194983 0.68 CA1 (0.47) CA9CA1CA2CA12
SCHEMBL27599728 0.67 PNMT (0.50)
SCHEMBL9301414 0.67 IDO1 (0.48) HPGDMEN1KMT2A
SCHEMBL10642950 0.66 PDIA6 (0.38) PTGES2CA9CA1CA2CA12
SCHEMBL10880283 0.65 FADS1 (0.46) HPGDHTTMEN1KMT2APTGS1
SCHEMBL24050785 0.65 CA2 (0.41) PTGES2CA9CA1CA2CA12
SCHEMBL5733314 0.65 PNMT (0.60)
SCHEMBL2436 0.65

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5314880-A Platelet activating factor antagonist BRITISH BIO-TECHNOLOGY LIMITED (GB) 1994-05-24 US disclosed
EP-0468971-A1 NOVEL BENZIMIDAZOLE DERIVATIVES BRITISH BIO-TECHNOLOGY LIMITED (GB) 1992-02-05 EP disclosed
WO-1990009997-A1 NOVEL BENZIMIDAZOLE DERIVATIVES BRITISH BIO-TECHNOLOGY LIMITED (GB) 1990-09-07 WO disclosed