SCHEMBL9301495

SCHEMBL9301495

COc1nc(N)c(N=O)c(=O)n1C

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 3/20 0.46
CCNA2 P20248 2/20 0.46
CCNA1 P78396 2/20 0.46
CASP6 P55212 2/20 0.42
CDK1 P06493 2/20 0.37
CDK4 P11802 1/20 0.37
RXFP1 Q9HBX9 1/20 0.36
CCNB1 P14635 1/20 0.32
KDM4E B2RXH2 1/20 0.30
MEN1 O00255 1/20 0.30
MAPT P10636 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9300537 0.78 DPP4 (0.32) KDM4EMEN1KMT2A
SCHEMBL9304641 0.74 CDK2 (0.39) CDK2CCNA2CCNA1CDK1CDK4
SCHEMBL8723623 0.72 RXFP1 (0.62) CDK2CCNA2CCNA1CASP6CDK1
SCHEMBL9663306 0.68 S100B (0.32) KDM4E
SCHEMBL17447368 0.66 CDK2 (0.70) CDK2CCNA2CCNA1CDK1CDK4
SCHEMBL16464949 0.63 CDK2 (1.00) CDK2CCNA2CCNA1CDK1CDK4
SCHEMBL22927782 0.62 TP53 (0.38) RXFP1KDM4EMEN1MAPTKMT2A
SCHEMBL4193697 0.62 CASP6 (0.66) CASP6RXFP1KDM4EMEN1MAPT
SCHEMBL28456121 0.61 KMT2A (0.60) RXFP1MEN1KMT2A
SCHEMBL14490772 0.60 CDK2 (0.47) CDK2CCNA2CCNA1CASP6CDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5314890-A Treatment of asthma MALESCI ISTITUTO FARMACOBIOLOGICO S.P.A. (IT) 1994-05-24 US disclosed
EP-0531349-A1 1-7 SUBSTITUTED XANTHINE DERIVATIVES HAVING ANTIASTHMATIC ACTIVITY, THEIR SALTS PHYSIOLOGICALLY ACCEPTABLE, PHARMACEUTICAL COMPOSITION CONTAINING THEM AND PROCESS FOR THEIR PREPARATION MALESCI ISTITUTO FARMACOBIOLOGICO S.p.A. (IT) 1993-03-17 EP disclosed
WO-1991017993-A1 1-7 SUBSTITUTED XANTHINE DERIVATIVES HAVING ANTIASTHMATIC ACTIVITY, THEIR SALTS PHYSIOLOGICALLY ACCEPTABLE, PHARMACEUTICAL COMPOSITION CONTAINING THEM AND PROCESS FOR THEIR PREPARATION MALESCI ISTITUTO FARMACOBIOLOGICO S.P.A (IT) 1991-11-28 WO disclosed