SCHEMBL9302340

SCHEMBL9302340

CCS(=O)(=O)NC(=O)c1cccc(N)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.57
ALDH1A1 P00352 2/20 0.57
SMN1; SMN2 Q16637 2/20 0.48
NPSR1 Q6W5P4 1/20 0.48
HSD17B10 Q99714 1/20 0.48
KDM4C Q9H3R0 1/20 0.47
PBRM1 Q86U86 1/20 0.46
KAT6A Q92794 1/20 0.46
PTGS1 P23219 1/20 0.44
LMNA P02545 2/20 0.44
NPC1 O15118 1/20 0.44
MITF O75030 1/20 0.44
POLB P06746 1/20 0.44
PRMT5 O14744 1/20 0.43
WDR77 Q9BQA1 1/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
ADRB2 P07550 1/20 0.43
ADRB1 P08588 1/20 0.43
ADRB3 P13945 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL478979 0.83 KDM4E (0.53) KDM4EALDH1A1SMN1; SMN2NPSR1HSD17B10
SCHEMBL7984974 0.82 L3MBTL1 (0.59) KDM4EALDH1A1SMN1; SMN2NPC1POLB
SCHEMBL7984819 0.82 HDAC8 (0.64) ALDH1A1SMN1; SMN2KAT6ANPC1POLB
Hydrochloric Acid SCHEMBL8306980 0.82 KDM4E (0.51) KDM4EALDH1A1SMN1; SMN2NPSR1HSD17B10
SCHEMBL17806411 0.81 SMN1; SMN2 (0.51) KDM4EALDH1A1SMN1; SMN2NPSR1HSD17B10
SCHEMBL7983790 0.81 HDAC1 (0.62) KDM4EALDH1A1SMN1; SMN2KAT6ALMNA
SCHEMBL7983817 0.81 FLT1 (0.61) ALDH1A1MEN1KMT2ACA1CA2
SCHEMBL29659751 0.81 HDAC1 (0.62) KDM4EALDH1A1SMN1; SMN2KAT6ALMNA
SCHEMBL24420690 0.80 LMNA (0.51) KDM4EALDH1A1SMN1; SMN2LMNANPC1
SCHEMBL8543957 0.79 ALDH1A1 (0.49) KDM4EALDH1A1SMN1; SMN2NPSR1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5360802-A Antagonists of cholecystokinin and gastrin MERCK SHARPE & DOHME LTD. 1994-11-01 US disclosed
EP-0514133-A1 Benzodiazepine derivatives, compositions containing them and their use in therapy MERCK SHARP & DOHME LTD. (GB) 1992-11-19 EP disclosed