SCHEMBL9302390

SCHEMBL9302390

COc1ccc(CSC[C@H](NC(=O)C(C)(C)SCc2ccc(OC)cc2)C(N)=O)cc1

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ACE P12821 5/20 0.51
PPARG P37231 4/20 0.51
PPARA Q07869 4/20 0.51
IDO1 P14902 2/20 0.44
EPHX1 P07099 1/20 0.44
GAA P10253 1/20 0.42
ALDH1A1 P00352 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
PKM P14618 1/20 0.39
PPARD Q03181 2/20 0.39
NPSR1 Q6W5P4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9301567 0.89 ACE (0.52) ACEPPARGPPARAGAAALDH1A1
SCHEMBL9301035 0.89 ACE (0.64) ACEPPARGPPARAPPARD
SCHEMBL4459598 0.84 ACE (0.56) ACEPPARGPPARAIDO1EPHX1
SCHEMBL9299216 0.76 PPARA (0.62) ACEPPARGPPARAEPHX1
SCHEMBL9299211 0.76 PPARA (0.62) ACEPPARGPPARAEPHX1
SCHEMBL11516592 0.75 ACE (0.60) ACEPPARGPPARAPPARD
SCHEMBL9848804 0.74 EPHX1 (0.53) ACEPPARGPPARAIDO1EPHX1
SCHEMBL9848809 0.74 EPHX1 (0.53) ACEPPARGPPARAIDO1EPHX1
SCHEMBL27360388 0.74 HTT (0.47) IDO1GAAALDH1A1SMN1; SMN2PKM
SCHEMBL6575981 0.73 MEN1 (0.54) ACEIDO1GAAALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5292926-A Cysteine derivatives SANTEN PHARMACEUTICAL CO., LTD. (JP) 1994-03-08 US disclosed
EP-0326326-A1 Cysteine derivatives SANTEN PHARMACEUTICAL CO., LTD. (JP) 1989-08-02 EP disclosed