SCHEMBL9302582

SCHEMBL9302582

CC(C)(C)OC(=O)N1CCN(c2cc3c(cc2F)n2c(=O)n(NC(=O)O)c(=O)cc2n3C2CC2)CC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.37
KDM4E B2RXH2 1/20 0.37
CDK4 P11802 1/20 0.36
CCND1 P24385 1/20 0.36
CCND2 P30279 1/20 0.36
CCND3 P30281 1/20 0.36
HRH3 Q9Y5N1 4/20 0.36
PIK3CA P42336 1/20 0.36
MTOR P42345 1/20 0.36
PRKDC P78527 1/20 0.36
OPRM1 P35372 1/20 0.35
OPRD1 P41143 1/20 0.35
OGFRL1 Q5TC84 1/20 0.35
TP53 P04637 2/20 0.35
MAPT P10636 2/20 0.35
LMNA P02545 1/20 0.35
THRB P10828 1/20 0.35
STS P08842 2/20 0.35
GPR119 Q8TDV5 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9303636 0.93 CDK4 (0.36) ALDH1A1KDM4ECDK4CCND1CCND2
SCHEMBL9303155 0.87 HRH3 (0.38) ALDH1A1KDM4ECDK4CCND1CCND2
SCHEMBL9303642 0.85 OPRM1 (0.36) ALDH1A1KDM4ECDK4CCND1CCND2
SCHEMBL9302286 0.85 OPRM1 (0.38) ALDH1A1KDM4ECDK4CCND1CCND2
SCHEMBL9301295 0.83 OPRM1 (0.36) ALDH1A1KDM4ECDK4CCND1CCND2
SCHEMBL9301342 0.83 STS (0.38) HRH3OPRM1OPRD1OGFRL1TP53
SCHEMBL9304073 0.80 MAPT (0.39) ALDH1A1KDM4EHRH3OPRM1OPRD1
SCHEMBL9302223 0.76 KDM4E (0.41) ALDH1A1KDM4EPIK3CAMAPTLMNA
SCHEMBL9847726 0.74 KDM4E (0.40) ALDH1A1KDM4EPIK3CAMAPTLMNA
SCHEMBL9301409 0.73 ALDH1A1 (0.41) ALDH1A1KDM4ETP53MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5283248-A Bactericides, enzyme inhibitor of DNA-gyrase in bacteria HOFFMANN-LA ROCHE INC. (US) 1994-02-01 US disclosed
EP-0433648-A1 Substituted pyrimidobenzimidazole derivatives F. HOFFMANN-LA ROCHE AG (CH) 1991-06-26 EP disclosed