SCHEMBL9304073

SCHEMBL9304073

CC(C)(C)OC(=O)N1CCN(c2cc3c(cc2F)n2c(=O)[nH]c(=O)cc2n3C2CC2)CC1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.39
KDM4E B2RXH2 3/20 0.39
THRB P10828 3/20 0.39
HRH3 Q9Y5N1 4/20 0.38
GPR119 Q8TDV5 2/20 0.38
OPRM1 P35372 1/20 0.38
OPRD1 P41143 1/20 0.38
OGFRL1 Q5TC84 1/20 0.38
ALDH1A1 P00352 3/20 0.37
TSHR P16473 2/20 0.37
POLB P06746 1/20 0.37
GAA P10253 1/20 0.37
HPGD P15428 1/20 0.37
ALOX15 P16050 1/20 0.37
HSD17B10 Q99714 1/20 0.37
DPP4 P27487 1/20 0.36
TP53 P04637 2/20 0.35
LMNA P02545 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9302040 0.87 KDM4E (0.41) MAPTKDM4EALDH1A1TSHRPOLB
SCHEMBL9302272 0.84 MAPT (0.42) MAPTKDM4ETHRBGPR119ALDH1A1
SCHEMBL9303155 0.84 HRH3 (0.38) MAPTKDM4ETHRBHRH3GPR119
SCHEMBL9302286 0.81 OPRM1 (0.38) MAPTKDM4ETHRBHRH3GPR119
SCHEMBL9301516 0.81 CASP3 (0.34) HRH3OPRM1OPRD1OGFRL1ALDH1A1
SCHEMBL9301445 0.80 ALDH1A1 (0.44) MAPTKDM4EALDH1A1TSHRGAA
SCHEMBL9303636 0.80 CDK4 (0.36) MAPTKDM4ETHRBHRH3GPR119
SCHEMBL9302582 0.80 ALDH1A1 (0.37) MAPTKDM4ETHRBHRH3GPR119
Trifluoroacetic Acid SCHEMBL9301612 0.80 KDM4E (0.46) MAPTKDM4EALDH1A1TSHRGAA
SCHEMBL9301295 0.79 OPRM1 (0.36) MAPTKDM4ETHRBHRH3GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5283248-A Bactericides, enzyme inhibitor of DNA-gyrase in bacteria HOFFMANN-LA ROCHE INC. (US) 1994-02-01 US disclosed