SCHEMBL9302844

SCHEMBL9302844

O=C(O)c1cc2cc(O)ccc2c(-c2ccccc2F)c1CO

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ACMSD Q8TDX5 1/20 0.42
GPR35 Q9HC97 4/20 0.41
SOS1 Q07889 2/20 0.41
LMNA P02545 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
CA12 O43570 1/20 0.39
CA9 Q16790 1/20 0.39
DHODH Q02127 5/20 0.38
POLB P06746 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
HCAR2 Q8TDS4 1/20 0.36
THRA P10827 1/20 0.36
THRB P10828 1/20 0.36
ESR1 P03372 1/20 0.36
ESR2 Q92731 1/20 0.36
HNF4A P41235 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9304643 0.85 THRA (0.44) GPR35SOS1CA12CA9POLB
SCHEMBL9242812 0.83 GRIN2D (0.44) GPR35SOS1POLBESR1ESR2
SCHEMBL9302889 0.80 ESR1 (0.41) GPR35SMN1; SMN2DHODHNPC1RAB9A
SCHEMBL9262474 0.76 POLB (0.41) GPR35SOS1POLBTHRBESR1
SCHEMBL9302205 0.75 ESR1 (0.44) GPR35CA12CA9DHODHNPC1
SCHEMBL9255419 0.74 ACMSD (0.44) ACMSDGPR35DHODH
SCHEMBL9255770 0.74 CYP3A4 (0.46) GPR35LMNASMN1; SMN2DHODH
SCHEMBL9303171 0.73 POLB (0.43) ACMSDGPR35SOS1POLBHCAR2
SCHEMBL9269222 0.73 HSD17B1 (0.42) GPR35SOS1CA12CA9POLB
SCHEMBL9302159 0.72 GPR35 (0.46) GPR35LMNASMN1; SMN2POLBNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5281720-A Antiasthmatics, antiallergens, antiinflammatory agents and cytoprotective agents MERCK FROSST CANADA, INC. 1994-01-25 US disclosed
US-5227399-A Pyranylphenyl naphthalene lactones as inhibitors of leukotriene biosynthesis MERCK FROSST CANADA, INC. (CA) 1993-07-13 US disclosed
EP-0501579-A1 Naphthalene lactones as inhibitors of leukotriene biosynthesis MERCK FROSST CANADA INC. (CA) 1992-09-02 EP disclosed
EP-0501578-A1 Pyranylphenyl hydroxyalkylnaphthoic acids as inhibitors of leukotriene biosynthesis MERCK FROSST CANADA INC. (CA) 1992-09-02 EP disclosed