SCHEMBL9302902

SCHEMBL9302902

COc1ccc(CCl)cc1C1CC(O)CCO1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TTR P02766 2/20 0.40
SIGMAR1 Q99720 1/20 0.38
CA1 P00915 4/20 0.36
CA2 P00918 4/20 0.36
CA9 Q16790 4/20 0.36
CA12 O43570 2/20 0.36
SLC5A1 P13866 1/20 0.36
SLC5A2 P31639 1/20 0.36
RECQL P46063 1/20 0.36
SLC6A2 P23975 3/20 0.35
SLC6A4 P31645 3/20 0.35
SLC6A3 Q01959 2/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
SELL P14151 1/20 0.35
SELP P16109 1/20 0.35
ATM Q13315 1/20 0.35
ACHE P22303 1/20 0.34
EP300 Q09472 2/20 0.34
ALDH1A1 P00352 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9303942 0.89 ACHE (0.45) SIGMAR1CA1CA2CA9CA12
SCHEMBL9301911 0.88 CA1 (0.39) SIGMAR1CA1CA2CA9CA12
SCHEMBL14244189 0.70 RECQL (0.60) TTRSIGMAR1RECQL
SCHEMBL20052995 0.69 POLL (0.37) SLC6A2SLC6A4MEN1KMT2A
SCHEMBL185845 0.67 CA2 (0.68) TTRSIGMAR1CA2ATMALDH1A1
SCHEMBL30074670 0.67 CA2 (0.68) TTRSIGMAR1CA2ATMALDH1A1
SCHEMBL5309679 0.67 PDE4B (0.56) RECQL
SCHEMBL20052948 0.66 ATM (0.42) CA1CA2CA9CA12ATM
SCHEMBL18856159 0.66 KDM4E (0.47) CA1CA2CA9CA12MEN1
SCHEMBL4976340 0.66 TTR (0.67) TTRCA2MEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5281720-A Antiasthmatics, antiallergens, antiinflammatory agents and cytoprotective agents MERCK FROSST CANADA, INC. 1994-01-25 US disclosed
US-5227399-A Pyranylphenyl naphthalene lactones as inhibitors of leukotriene biosynthesis MERCK FROSST CANADA, INC. (CA) 1993-07-13 US disclosed
EP-0501579-A1 Naphthalene lactones as inhibitors of leukotriene biosynthesis MERCK FROSST CANADA INC. (CA) 1992-09-02 EP disclosed
EP-0501578-A1 Pyranylphenyl hydroxyalkylnaphthoic acids as inhibitors of leukotriene biosynthesis MERCK FROSST CANADA INC. (CA) 1992-09-02 EP disclosed