SCHEMBL9303314

SCHEMBL9303314

CC[Si](CC)(CCc1cc(CC(C)C)c(O)c(CC(C)C)c1)CCc1cc(CC(C)C)c(O)c(CC(C)C)c1

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 2/20 0.43
GABRB2 P47870 2/20 0.43
ALOX5 P09917 1/20 0.31
NFKB1 P19838 1/20 0.31
NFKB2 Q00653 1/20 0.31
RELA Q04206 1/20 0.31
ALOX15 P16050 1/20 0.30
ALOX12 P18054 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9194816 0.86 GABRA1 (0.40) GABRA1GABRB2
SCHEMBL5692470 0.83 GABRA1 (0.46) GABRA1GABRB2ALOX5NFKB1NFKB2
SCHEMBL9193711 0.83 GABRA1 (0.46) GABRA1GABRB2ALOX5NFKB1NFKB2
SCHEMBL9193282 0.81 DHFR (0.41) GABRA1GABRB2ALOX5
SCHEMBL16182674 0.80 GABRA1 (0.50) GABRA1GABRB2ALOX5NFKB1NFKB2
SCHEMBL9192781 0.78 HTT (0.42) GABRA1GABRB2ALOX5ALOX15
SCHEMBL4659133 0.77 NPC1 (0.48) GABRA1GABRB2
SCHEMBL8342795 0.76 GABRA1 (0.54) GABRA1GABRB2NFKB1ALOX15ALOX12
SCHEMBL28720288 0.76 PTGS2 (0.53) GABRA1GABRB2
SCHEMBL9195415 0.76 GABRA1 (0.51) GABRA1GABRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5304668-A Bis-[4-(2,6-di-alkyl)phenolisilane derivatives as antiatherosclerotic agents MERRELL DOW PHARMACEUTICALS (US) 1994-04-19 US disclosed
US-5281738-A Anticholesterol agents MERRELL DOW PHARMACEUTICALS INC. (US) 1994-01-25 US disclosed