SCHEMBL9303930

SCHEMBL9303930

O=C=Nc1ccc(Br)c2c(N=C=O)ccc(Br)c12

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.41
TDP1 Q9NUW8 2/20 0.38
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
TRPA1 O75762 1/20 0.36
TSHR P16473 1/20 0.32
GABRA1 P14867 1/20 0.30
GABRB2 P47870 1/20 0.30
MAPK1 P28482 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4285629 0.79 CYP3A4 (0.40) CYP3A4TDP1ALDH1A1HPGDTRPA1
SCHEMBL9304725 0.76 ALDH1A1 (0.38) CYP3A4TDP1ALDH1A1HPGD
SCHEMBL11601249 0.76 CYP3A4 (0.38) CYP3A4TDP1ALDH1A1HPGDTRPA1
SCHEMBL17847475 0.74 CYP3A4 (0.45) CYP3A4TDP1ALDH1A1HPGDTRPA1
SCHEMBL5786288 0.74 CYP3A4 (0.41) CYP3A4TDP1ALDH1A1HPGDTRPA1
SCHEMBL2156211 0.73 CYP3A4 (0.53) CYP3A4TDP1ALDH1A1HPGDTRPA1
SCHEMBL1457695 0.73 HSP90AA1 (0.41) CYP3A4TDP1ALDH1A1HPGDTRPA1
SCHEMBL93220 0.71 CYP3A4 (0.52) CYP3A4TDP1ALDH1A1HPGDTRPA1
SCHEMBL29463737 0.71 CYP3A4 (0.52) CYP3A4TDP1ALDH1A1HPGDTRPA1
SCHEMBL9630369 0.71 CYP3A4 (0.55) CYP3A4TDP1ALDH1A1HPGDTRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5349062-A Charge tranfer compounds CIBA-GEIGY CORPORATION (US) 1994-09-20 US disclosed
EP-0577560-A1 Substituted naphtho[1,8-de:5,4-d'e']bis[1,3]thiazines, process for their preparation and their electrically conductive charge transfer complexes CIBA-GEIGY AG (CH) 1994-01-05 EP disclosed