SCHEMBL9307764

SCHEMBL9307764

CCCCCCCCCCCCCCOc1ccc(NCc2cccnc2)cc1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.58
LTA4H P09960 1/20 0.55
TSHR P16473 2/20 0.54
CYP3A4 P08684 2/20 0.53
CYP2D6 P10635 2/20 0.53
CYP2C9 P11712 2/20 0.53
CYP2C19 P33261 2/20 0.53
CYP19A1 P11511 1/20 0.53
POLB P06746 2/20 0.53
TP53 P04637 1/20 0.53
TDP1 Q9NUW8 1/20 0.53
NFKB1 P19838 2/20 0.53
NFKB2 Q00653 2/20 0.53
RELA Q04206 2/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
NPC1 O15118 1/20 0.53
MAPT P10636 1/20 0.53
LMNA P02545 1/20 0.53
GAA P10253 1/20 0.51
FAAH O00519 7/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23873637 0.85 ALDH1A1 (0.72) ALDH1A1LTA4HCYP3A4CYP2D6CYP2C9
SCHEMBL855997 0.84 CACNA1B (0.58) LTA4HTP53MAPTGAAFAAH
SCHEMBL2908596 0.79 ALDH1A1 (0.69) ALDH1A1LTA4HCYP3A4CYP2D6CYP2C9
SCHEMBL9309140 0.78 CACNA1B (0.58) LTA4HTP53MAPTGAAFAAH
SCHEMBL6394149 0.77 CACNA1B (0.50) ALDH1A1CYP3A4SMN1; SMN2NPC1LMNA
SCHEMBL10556321 0.76 LTA4H (0.57) ALDH1A1LTA4HCYP3A4CYP2D6CYP2C9
SCHEMBL13766317 0.76 ALDH1A1 (0.73) ALDH1A1LTA4HCYP3A4CYP2D6CYP2C9
SCHEMBL9164953 0.76 NR5A1 (0.51) ALDH1A1CYP3A4SMN1; SMN2NPC1LMNA
SCHEMBL4888697 0.76 CHRNB2 (0.62) LTA4HTSHRCYP3A4CYP2D6CYP2C9
SCHEMBL9367178 0.76 CHRNB2 (0.62) LTA4HTSHRCYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5328921-A Antagonist of platelet activating factor AMERICAN CYANAMID COMPANY (US) 1994-07-12 US disclosed
US-5208247-A Antianaphylactic agents or septic shock AMERICAN CYANAMID COMPANY (US) 1993-05-04 US disclosed
EP-0530444-A1 Aryl, amide, imide, and carbamate pyridine antagonists of platelet activating factor AMERICAN CYANAMID COMPANY (US) 1993-03-10 EP disclosed