SCHEMBL932679

SCHEMBL932679

COc1ccc(C2(C3CC4CCC3C4)N=C(C)C(N)=N2)cc1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 9/20 0.41
KCNH2 Q12809 2/20 0.41
PRMT5 O14744 3/20 0.36
CTSD P07339 3/20 0.36
WDR77 Q9BQA1 3/20 0.36
BACE2 Q9Y5Z0 2/20 0.36
REN P00797 1/20 0.36
CYP3A4 P08684 1/20 0.35
CTSE P14091 1/20 0.35
CYP2C19 P33261 1/20 0.35
MAOB P27338 2/20 0.34
MAOA P21397 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL932399 0.76 BACE1 (0.53) BACE1KCNH2BACE2CYP3A4CTSE
SCHEMBL931327 0.76 BACE1 (0.53) BACE1KCNH2BACE2CYP3A4CTSE
SCHEMBL931861 0.76 BACE1 (0.53) BACE1KCNH2BACE2CYP3A4CTSE
SCHEMBL3686002 0.61 KDM1A (0.55) MAOBMAOA
SCHEMBL931601 0.61 BACE1 (0.50) BACE1KCNH2BACE2
SCHEMBL6922254 0.58 BACE1 (0.69) BACE1KCNH2CTSDBACE2
SCHEMBL932572 0.58 BACE1 (0.69) BACE1KCNH2CTSDBACE2
SCHEMBL21895378 0.58 FABP7 (0.46) CYP3A4
SCHEMBL8766773 0.57 HSD11B1 (0.56) BACE1PRMT5CTSDWDR77BACE2
SCHEMBL14667567 0.57 ALDH1A1 (0.54) CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011002408-A1 NOVEL COMPOUNDS FOR TREATMENT OF NEURODEGENERATION ASSOCIATED WITH DISEASES, SUCH AS ALZHEIMER'S DISEASE OR DEMENTIA ASTRAZENECA AB (SE) 2011-01-06 WO disclosed
WO-2011002408-A1 NOVEL COMPOUNDS FOR TREATMENT OF NEURODEGENERATION ASSOCIATED WITH DISEASES, SUCH AS ALZHEIMER'S DISEASE OR DEMENTIA ASTRAZENECA AB (SE) 2011-01-06 WO disclosed