SCHEMBL9313614

SCHEMBL9313614

N#Cc1ccccc1-c1cccc2c(CBr)cccc12

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.40
MAPT P10636 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
ESR2 Q92731 1/20 0.40
TSHR P16473 2/20 0.35
DYRK1A Q13627 2/20 0.34
CYP19A1 P11511 2/20 0.34
IMPDH2 P12268 1/20 0.33
IMPDH1 P20839 1/20 0.33
CNR2 P34972 1/20 0.33
MCL1 Q07820 1/20 0.33
CYP1A1 P04798 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP1B1 Q16678 1/20 0.33
PTGES O14684 1/20 0.33
GALR3 O60755 1/20 0.33
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL588692 0.85 ESR2 (0.44) ALDH1A1MAPTSMN1; SMN2ESR2TSHR
SCHEMBL2940694 0.85 SLC6A2 (0.42) ALDH1A1MAPTSMN1; SMN2CA1CA2
SCHEMBL20631601 0.84 ALDH1A1 (0.42) ALDH1A1MAPTSMN1; SMN2CA1CA2
SCHEMBL3644296 0.83 ESR2 (0.40) ALDH1A1MAPTSMN1; SMN2CA1CA2
SCHEMBL2575065 0.81 GABRA1 (0.39) CA1CA2ESR2TSHRCYP19A1
SCHEMBL2462113 0.78 CYP19A1 (0.50) ALDH1A1MAPTSMN1; SMN2CA1CA2
SCHEMBL29559172 0.78 CYP19A1 (0.50) ALDH1A1MAPTSMN1; SMN2CA1CA2
SCHEMBL899 0.77 CYP19A1 (0.46) ALDH1A1MAPTSMN1; SMN2CA1CA2
SCHEMBL29513232 0.77 CYP19A1 (0.46) ALDH1A1MAPTSMN1; SMN2CA1CA2
SCHEMBL28203557 0.76 CA1 (0.60) ALDH1A1CA1CA2ESR2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5350752-A Dihydropyrimidine derivatives E. R. SQUIBB & SONS, INC. (US) 1994-09-27 US disclosed
EP-0547442-A1 Dihydropyrimidin derivatives used as A-II receptor antagonists E.R. SQUIBB & SONS, INC. (US) 1993-06-23 EP disclosed