SCHEMBL9316280

SCHEMBL9316280

Cc1cc(Br)ccc1N=C(NNC(=Nc1ccc(Br)cc1C)NC12CC3CC(CC(C3)C1)C2)NC1CCCCC1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 6/20 0.40
EPHX1 P07099 2/20 0.40
SIGMAR1 Q99720 3/20 0.36
TSHR P16473 1/20 0.35
KDM4E B2RXH2 1/20 0.35
NPC1 O15118 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
CNR2 P34972 2/20 0.34
MAPT P10636 1/20 0.34
FAAH O00519 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9316291 0.90 EPHX2 (0.33) EPHX2EPHX1CNR2FAAH
SCHEMBL9317615 0.84 SIGMAR1 (0.45) EPHX2EPHX1SIGMAR1TSHRNPC1
SCHEMBL8952180 0.77 SIGMAR1 (0.53) EPHX2SIGMAR1KDM4ENPC1ALDH1A1
SCHEMBL6719600 0.76 SIGMAR1 (0.54) EPHX2SIGMAR1KDM4ENPC1ALDH1A1
SCHEMBL9316317 0.75 RAC1 (0.39) EPHX2EPHX1SIGMAR1MAPT
SCHEMBL8952043 0.74 SIGMAR1 (0.56) EPHX1SIGMAR1NPC1ALDH1A1LMNA
SCHEMBL8952040 0.74 SIGMAR1 (0.56) EPHX1SIGMAR1NPC1ALDH1A1LMNA
SCHEMBL6719371 0.73 SIGMAR1 (0.57) EPHX2EPHX1SIGMAR1NPC1ALDH1A1
SCHEMBL8741839 0.71 TAS1R3 (0.49) EPHX1SIGMAR1NPC1LMNARAB9A
SCHEMBL8952184 0.67 SIGMAR1 (0.44) EPHX2SIGMAR1KDM4ENPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0532642-A4 1994-04-27 EP disclosed
EP-0532642-A1 SUBSTITUTED GUANIDINES HAVING HIGH BINDING TO THE SIGMA RECEPTOR AND THE USE THEREOF STATE OF OREGON, acting through OREGON STATE BOARD OF HIGHER EDUCATION, acting for OREGON HEALTH SC. UNIV. AND UNIV. OF OREGON (US) 1993-03-24 EP disclosed
WO-1991018868-A1 SUBSTITUTED GUANIDINES HAVING HIGH BINDING TO THE SIGMA RECEPTOR AND THE USE THEREOF STATE OF OREGON, acting by and through the OREGON STATE BOARD OF HIGHER EDUCATION, acting for and onbehalf of the OREGON HEALTH SCIENCES UNIVERSITY (US) 1991-12-12 WO disclosed