SCHEMBL9316462

SCHEMBL9316462

O=C(O)c1c(N2Cc3cccnc3C2)n(C2CC2)c2ncc(F)cc2c1=O

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TIPARP Q7Z3E1 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
PIK3CG P48736 1/20 0.33
TLR2 O60603 1/20 0.33
AOC3 Q16853 1/20 0.32
ELANE P08246 1/20 0.31
TOP2A P11388 1/20 0.31
TOP2B Q02880 1/20 0.31
IRAK4 Q9NWZ3 1/20 0.31
NAMPT P43490 1/20 0.31
PIK3CA P42336 2/20 0.31
RIPK1 Q13546 1/20 0.31
PDE4B Q07343 2/20 0.30
PDE4D Q08499 2/20 0.30
PDE4A P27815 1/20 0.30
PDE4C Q08493 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
HTR3A P46098 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9651894 0.88 HDAC6 (0.35) TIPARPHDAC6PIK3CGAOC3PDE4B
SCHEMBL9844933 0.74 HTR3A (0.33) PIK3CACYP1A2CYP3A4HTR3A
SCHEMBL30954833 0.73 NAMPT (0.37) TIPARPAOC3IRAK4NAMPT
SCHEMBL27291990 0.70 ELANE (0.40) ELANETOP2ATOP2BPDE4BPDE4D
SCHEMBL6530640 0.69 KCNH2 (0.37)
SCHEMBL9316471 0.67 PIK3CG (0.65) PIK3CGTOP2ATOP2BPIK3CACYP1A2
SCHEMBL10594808 0.66 CYP11B2 (0.35) TOP2ATOP2BCYP1A2CYP3A4HTR3A
SCHEMBL9317503 0.66 TOP2A (0.57) PIK3CGTOP2ATOP2B
SCHEMBL8589216 0.65 ELANE (0.42) ELANEPIK3CAPDE4BPDE4D
SCHEMBL27283744 0.65 DDB1 (0.40) ELANEPDE4BPDE4DPDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5371090-A Bactericides, feed additives BAYER AKTIENGESELLSCHAFT (DE) 1994-12-06 US disclosed
US-5312823-A Antibacterials BAYER AKTIENGESELLSCHAFT (DE) 1994-05-17 US disclosed
CN-1068114-A 7-azepine iso-dihydro-indole-group-quinolone and naphthyridonecarboxylic derivative BAYER AG (DE) 1993-01-20 CN disclosed