SCHEMBL9317620

SCHEMBL9317620

O=C(O)CCNC(=O)c1cc(I)ccc1Nc1ccc(C(F)(F)F)cc1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.47
AKR1C2 P52895 1/20 0.47
EPHX2 P34913 2/20 0.46
GCGR P47871 6/20 0.44
TRPV1 Q8NER1 2/20 0.43
PPARA Q07869 3/20 0.41
HSPH1 Q92598 1/20 0.41
PPARG P37231 2/20 0.40
RXFP1 Q9HBX9 1/20 0.40
PPARD Q03181 1/20 0.39
NR1H4 Q96RI1 1/20 0.39
FFAR1 O14842 1/20 0.39
MAP2K2 P36507 1/20 0.39
MAP2K1 Q02750 1/20 0.39
FBP1 P09467 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7332598 0.85 AKR1C3 (0.43) AKR1C3AKR1C2TRPV1PPARAPPARD
SCHEMBL9317706 0.85 GCG (0.44) AKR1C3AKR1C2GCGRMAP2K2MAP2K1
SCHEMBL9318985 0.82 AKR1C3 (0.48) AKR1C3AKR1C2
SCHEMBL8959409 0.76 NPSR1 (0.40) PPARAPPARGNR1H4MAP2K2MAP2K1
SCHEMBL7322396 0.72 ALDH1A1 (0.45) AKR1C3AKR1C2
SCHEMBL5782704 0.71 SIRT5 (0.53) EPHX2GCGRPPARA
SCHEMBL7330066 0.71 KCNQ2 (0.47) EPHX2PPARAPPARGPPARD
SCHEMBL7329535 0.71 CA1 (0.42)
SCHEMBL7326028 0.70 MAPT (0.41) AKR1C3AKR1C2
SCHEMBL7325535 0.70 MAPT (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0610334-A1 NONPEPTIDYL INTEGRIN INHIBITORS HAVING SPECIFICITY FOR THE GPII b?III a? RECEPTOR. GENENTECH INC (US) 1994-08-17 EP disclosed