SCHEMBL932044

SCHEMBL932044

O=CCN1CCc2cc(CCBr)ccc21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 1/20 0.39
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
ALDH1A1 P00352 2/20 0.34
LMNA P02545 2/20 0.34
KDM4E B2RXH2 2/20 0.34
TP53 P04637 2/20 0.34
MAPT P10636 2/20 0.34
GAA P10253 1/20 0.34
CASP1 P29466 1/20 0.34
HTT P42858 1/20 0.34
CASP7 P55210 1/20 0.34
SMAD3 P84022 1/20 0.34
HSD17B10 Q99714 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
HDAC1 Q13547 2/20 0.33
HDAC8 Q9BY41 2/20 0.33
HDAC6 Q9UBN7 2/20 0.33
USP2 O75604 1/20 0.33
CDK4 P11802 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL931550 0.86 S1PR1 (0.42) S1PR1MEN1KMT2AALDH1A1LMNA
SCHEMBL931075 0.79 SIGMAR1 (0.48) S1PR1HTR2CHTR2B
SCHEMBL9901142 0.79 HDAC1 (0.43) MEN1KMT2AALDH1A1LMNAMAPT
SCHEMBL16370572 0.76 ATAD2 (0.44) S1PR1MEN1KMT2AALDH1A1KDM4E
SCHEMBL14473300 0.74 ALDH1A1 (0.44) MEN1KMT2AALDH1A1LMNAKDM4E
SCHEMBL14473305 0.74 ALDH1A1 (0.50) MEN1KMT2AALDH1A1LMNAKDM4E
SCHEMBL466270 0.72 ALDH1A1 (0.63) MEN1KMT2AALDH1A1LMNAKDM4E
SCHEMBL1867023 0.71 MAPT (0.45) KMT2AALDH1A1LMNAMAPTGAA
SCHEMBL3783835 0.71 NOTUM (0.60) ALDH1A1LMNAKDM4ETP53MAPT
SCHEMBL2594028 0.71 CA1 (0.50) MEN1KMT2AALDH1A1KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2448934-A1 2-CARBOXAMIDE-7-PIPERAZINYL-BENZOFURAN DERIVATIVES 774 AstraZeneca AB (SE) 2012-05-09 EP disclosed
WO-2011002405-A1 2-CARBOXAMIDE-7-PIPERAZINYL-BENZOFURAN DERIVATIVES 774 ASTRAZENECA AB (SE) 2011-01-06 WO disclosed