SCHEMBL9320653

SCHEMBL9320653

CS(=O)(=O)O.O=C(OO)c1ccncc1

nearest known ligand 0.50

Known targets — ChEMBL curated mechanism

ABL1ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB2AGTR1BCL2BCL2A1BCL2L1BCL2L10BCL2L2BCRBRAFCHRM1CHRNA10CHRNA9DRD1DRD2DRD3DRD4DRD5EGFRF2FLT1FLT4GCKGHSRGNRHRGRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BHTR1AHTR1BHTR1DHTR2AHTR2CHTR3AIDH2KDRKITMAOBMCL1MTTPPP4HBPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PIKFYVEROCK1ROCK2SLC18A2SLC6A2SLC6A3SLC6A4TACR1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8gyrAgyrBparCparEpol

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 1/20 0.50
HPGD P15428 1/20 0.47
CYP1A2 P05177 2/20 0.47
CYP2C19 P33261 2/20 0.47
LMNA P02545 1/20 0.47
CYP2C9 P11712 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
HTT P42858 1/20 0.47
PTGS2 P35354 2/20 0.46
POLB P06746 2/20 0.46
LTA4H P09960 1/20 0.46
ALDH1A1 P00352 1/20 0.45
MAPT P10636 2/20 0.44
NAPRT Q6XQN6 1/20 0.43
TP53 P04637 1/20 0.43
KDM4E B2RXH2 1/20 0.42
MPO P05164 1/20 0.42
CYP3A4 P08684 1/20 0.42
ADORA3 P0DMS8 1/20 0.42
CYP2D6 P10635 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21397880 0.88 HSD17B10 (0.61) HSD17B10CYP1A2CYP2C19LMNACYP2C9
SCHEMBL31501741 0.80 CYP3A4 (0.50) HSD17B10HPGDCYP1A2CYP2C19CYP2C9
SCHEMBL9318729 0.79 ALDH1A1 (0.67) CYP1A2LMNACYP2C9PTGS2ALDH1A1
Methyl Isonicotinate SCHEMBL180574 0.77 CYP1A2 (0.60) HSD17B10CYP1A2CYP2C19LMNACYP2C9
Methyl Isonicotinate SCHEMBL820082 0.77 CYP1A2 (0.60) HSD17B10CYP1A2CYP2C19LMNACYP2C9
SCHEMBL9318493 0.77 ATM (0.50) CYP1A2CYP2C19CYP2C9PTGS2ALDH1A1
SCHEMBL27592050 0.76 HSD17B10 (0.53) HSD17B10HPGDCYP1A2CYP2C19LMNA
Methyl Isonicotinate SCHEMBL9213497 0.75 LMNA (0.58) HSD17B10CYP1A2CYP2C19LMNACYP2C9
Methyl Isonicotinate SCHEMBL9217491 0.75 LMNA (0.58) HSD17B10CYP1A2CYP2C19LMNACYP2C9
Methyl Isonicotinate SCHEMBL29827431 0.75 LMNA (0.58) HSD17B10CYP1A2CYP2C19LMNACYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0300461-B1 Aromatic heterocyclic peroxyacids AUSIMONT SPA (IT) 1994-01-12 EP claimed
US-4902803-A Aromatic heterocyclic peroxycarboxylic acids AUSIMONT S.P.A. (IT) 1990-02-20 US claimed
EP-0300461-A2 Aromatic heterocyclic peroxyacids AUSIMONT S.p.A. (IT) 1989-01-25 EP claimed
EP-0300461-B1 Aromatic heterocyclic peroxyacids AUSIMONT SPA (IT) 1994-01-12 EP disclosed
US-4902803-A Aromatic heterocyclic peroxycarboxylic acids AUSIMONT S.P.A. (IT) 1990-02-20 US disclosed
EP-0300461-A2 Aromatic heterocyclic peroxyacids AUSIMONT S.p.A. (IT) 1989-01-25 EP disclosed