SCHEMBL9320971

SCHEMBL9320971

CCCCCCCCCCCCCCCCC=CN(Cc1ccc(OCCN)c(OC)c1)C(=O)O

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 3/20 0.47
PTGER3 P43115 1/20 0.47
EPHX2 P34913 1/20 0.46
HTR1A P08908 3/20 0.44
TRPV1 Q8NER1 3/20 0.42
CYP1A2 P05177 2/20 0.42
CYP3A4 P08684 2/20 0.42
CYP2D6 P10635 2/20 0.42
THRA P10827 1/20 0.42
THRB P10828 1/20 0.42
CYP2E1 P05181 1/20 0.42
ALOX5 P09917 1/20 0.42
CYP2C8 P10632 1/20 0.42
CYP2A6 P11509 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2B6 P20813 1/20 0.42
CYP2C19 P33261 1/20 0.42
S1PR2 O95136 1/20 0.42
S1PR1 P21453 1/20 0.42
S1PR3 Q99500 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9320976 0.91 LTA4H (0.42) LTA4HPTGER3EPHX2HTR1AS1PR2
SCHEMBL9320967 0.86 EPHX2 (0.47) LTA4HPTGER3EPHX2HTR1ATRPV1
SCHEMBL9321717 0.81 THRA (0.47) PTGER3THRATHRBS1PR2S1PR1
SCHEMBL9320996 0.81 THRA (0.47) PTGER3THRATHRBS1PR2S1PR1
SCHEMBL9320972 0.80 EPHX2 (0.43) LTA4HPTGER3EPHX2THRATHRB
SCHEMBL9321037 0.79 EPHX2 (0.57) EPHX2TRPV1CYP1A2CYP3A4CYP2D6
SCHEMBL9321046 0.79 EPHX2 (0.57) EPHX2TRPV1CYP1A2CYP3A4CYP2D6
SCHEMBL9321040 0.78 FAAH (0.65) EPHX2TRPV1CYP1A2CYP3A4CYP2D6
SCHEMBL9321739 0.78 EPHX2 (0.51) LTA4HEPHX2TRPV1CYP1A2CYP3A4
SCHEMBL6700457 0.78 EPHX2 (0.51) LTA4HEPHX2TRPV1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0282127-B1 Beta-aminoethyl-substituted phenyl compounds, and anti-inflammatory or analgesic compositions containing them PROCTER & GAMBLE (US) 1994-02-02 EP disclosed
US-5099030-A Phenols or phenolic ethers THE PROCTER & GAMBLE COMPANY (US) 1992-03-24 US disclosed
US-5045565-A Novel compounds, pharmaceutical compositions, and methods for treating inflammation and pain THE PROCTER & GAMBLE COMPANY (US) 1991-09-03 US disclosed
EP-0282127-A2 Beta-aminoethyl-substituted phenyl compounds, and anti-inflammatory or analgesic compositions containing them THE PROCTER & GAMBLE COMPANY (US) 1988-09-14 EP disclosed