SCHEMBL9321672

SCHEMBL9321672

O=[C]c1ccccc1NC(=O)C(F)(F)F

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 8/20 0.51
PDK2 Q15119 8/20 0.51
PDK3 Q15120 8/20 0.51
PDK4 Q16654 8/20 0.51
TP53 P04637 2/20 0.49
JAK2 O60674 1/20 0.49
MAPT P10636 1/20 0.49
HTT P42858 1/20 0.49
KLK7 P49862 1/20 0.49
PARP14 Q460N5 1/20 0.43
MEN1 O00255 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
KMT2A Q03164 1/20 0.41
HSD17B10 Q99714 1/20 0.41
HDAC1 Q13547 2/20 0.40
HDAC7 Q8WUI4 2/20 0.40
HDAC8 Q9BY41 2/20 0.40
HDAC6 Q9UBN7 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20821412 0.84 PDK1 (0.50) PDK1PDK2PDK3PDK4TP53
SCHEMBL1542594 0.84 PDK1 (0.50) PDK1PDK2PDK3PDK4TP53
SCHEMBL4344024 0.84 PDK1 (0.70) PDK1PDK2PDK3PDK4TP53
SCHEMBL29824473 0.84 PDK1 (0.50) PDK1PDK2PDK3PDK4TP53
SCHEMBL14448754 0.81 PDK1 (0.51) PDK1PDK2PDK3PDK4TP53
SCHEMBL28528551 0.80 ALDH1A1 (0.58) PDK1PDK2PDK3PDK4TP53
SCHEMBL8626954 0.78 PDK1 (0.66) PDK1PDK2PDK3PDK4MAPT
SCHEMBL12758952 0.77 PDK1 (0.44) PDK1PDK2PDK3PDK4TP53
SCHEMBL1576313 0.76 PDK1 (0.67) PDK1PDK2PDK3PDK4TP53
SCHEMBL553679 0.76 ALDH1A1 (0.57) HTTMEN1NPC1RAB9AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5369123-A Anticholesterol agents, treatment of atherosclerosis, antilipidemic agents and treatment of hyperlipoproteinaemia E. R. SQUIBB & SONS, INC. (US) 1994-11-29 US disclosed