SCHEMBL932694

SCHEMBL932694

Cc1ccc(-c2nc(C#N)n(S(=O)(=O)N(C)C)c2Cl)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
ERBB2 P04626 1/20 0.38
TSHR P16473 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
ADORA1 P30542 4/20 0.35
ADORA2A P29274 2/20 0.35
MYC P01106 1/20 0.34
WDR5 P61964 1/20 0.34
KDM1A O60341 1/20 0.34
MEN1 O00255 2/20 0.33
PTGS2 P35354 2/20 0.33
ADORA2B P29275 1/20 0.33
HTT P42858 1/20 0.33
ALDH1A1 P00352 2/20 0.33
LMNA P02545 1/20 0.33
POLB P06746 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9520829 0.91 PTGS2 (0.39) KMT2ACYP1A2CYP2C9CYP2C19ERBB2
SCHEMBL9323989 0.88 TSHR (0.49) KMT2ACYP1A2CYP2C9CYP2C19ERBB2
SCHEMBL933896 0.88 ADORA1 (0.42) KMT2ATSHRSMN1; SMN2ADORA1ADORA2A
SCHEMBL933331 0.86 TSHR (0.34) KMT2ATSHRSMN1; SMN2PTGS2LMNA
SCHEMBL4858808 0.85 CYP1A2 (0.36) KMT2ACYP1A2CYP2C9CYP2C19ERBB2
Cyazofamid SCHEMBL22923 0.82 PTGS2 (0.38) KMT2ACYP1A2CYP2C9CYP2C19ERBB2
Cyazofamid SCHEMBL16180421 0.82 PTGS2 (0.38) KMT2ACYP1A2CYP2C9CYP2C19ERBB2
SCHEMBL932277 0.82 PTGS2 (0.39) TSHRPTGS2HTTALDH1A1LMNA
Cyazofamid SCHEMBL23804496 0.80 PTGS2 (0.37) KMT2ACYP1A2CYP2C9CYP2C19ERBB2
SCHEMBL9519745 0.76 SMN1; SMN2 (0.33) SMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 83 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0973397-A1 NOVEL FUNGICIDE COMPOSITION CONTAINING A 2-IMIDAZOLINE-5-ONE RHONE-POULENC AGROCHIMIE (FR) 2000-01-26 EP claimed
WO-1999027788-A1 NOVEL FUNGICIDE COMPOSITION CONTAINING A 2-IMIDAZOLINE-5-ONE RHONE POULENC AGROCHIMIE (FR) 1999-06-10 WO claimed
EP-2663188-A1 METHOD FOR CONTROLLING CLUBROOT Ishihara Sangyo Kaisha, Ltd. (JP) 2013-11-20 EP disclosed
WO-2012096405-A1 METHOD FOR CONTROLLING CLUBROOT ISHIHARA SANGYO KAISHA, LTD. (JP) 2012-07-19 WO disclosed
EP-2451275-A1 AGRICULTURAL OR HORTICULTURAL FUNGICIDE COMPOSITION AND ITS USE FOR CONTROLLING PLANT PATHOGENS Ishihara Sangyo Kaisha, Ltd. (JP) 2012-05-16 EP disclosed
EP-2320733-A2 METHOD FOR CONTROLLING DEGRADATION OF AGRICULTURAL CHEMICAL ACTIVE INGREDIENT ISHIHARA SANGYO KAISHA, LTD. (JP) 2011-05-18 EP disclosed
WO-2011004901-A1 AGRICULTURAL OR HORTICULTURAL FUNGICIDE COMPOSITION AND ITS USE FOR CONTROLLING PLANT PATHOGENS ISHIHARA SANGYO KAISHA, LTD. (JP) 2011-01-13 WO disclosed
WO-2010021404-A2 METHOD FOR CONTROLLING DEGRADATION OF AGRICULTURAL CHEMICAL ACTIVE INGREDIENT ISHIHARA SANGYO KAISHA, LTD. (JP) 2010-02-25 WO disclosed
EP-1504001-B1 2-(2-PYRIDYL)-5-PHENYL-6-AMINOPYRIMIDINE, METHOD AND INTERMEDIATE PRODUCTS FOR THE PRODUCTION AND USE THEREOF FOR COMBATING NOXIOUS FUNGI BASF SE (DE) 2009-04-15 EP disclosed
US-7320975-B2 2-(2-pyridyl)-5-phenyl-6-aminopyrimidine, method and intermediate products for the production and use thereof for combating noxious fungi BASF AKTIENGESELLSCHAFT (DE) 2008-01-22 US disclosed
EP-1490372-B1 FUNGICIDAL TRIAZOLOPYRIMIDINES, METHODS FOR PRODUCING THE SAME, USE THEREOF FOR COMBATING HARMFUL FUNGI AND AGENTS CONTAINING SAID SUBSTANCES BASF AG (DE) 2008-01-16 EP disclosed
EP-1194039-A2 PESTICIDAL COMPOSITION AND METHOD FOR CONTROLLING PESTS ISHIHARA SANGYO KAISHA, LTD. (JP) 2002-04-10 EP disclosed
WO-2001005231-A2 PESTICIDAL COMPOSITION AND METHOD FOR CONTROLLING PESTS ISHIHARA SANGYO KAISHA, LTD. (JP) 2001-01-25 WO disclosed
EP-0979034-A1 COMPOSITION FOR CONTROLLING HARMFUL BIO-ORGANISMS AND METHOD FOR CONTROLLING HARMFUL BIO-ORGANISMS USING THE SAME ISHIHARA SANGYO KAISHA, LTD. (JP) 2000-02-16 EP disclosed
EP-0973397-A1 NOVEL FUNGICIDE COMPOSITION CONTAINING A 2-IMIDAZOLINE-5-ONE RHONE-POULENC AGROCHIMIE (FR) 2000-01-26 EP disclosed
WO-1999027788-A1 NOVEL FUNGICIDE COMPOSITION CONTAINING A 2-IMIDAZOLINE-5-ONE RHONE POULENC AGROCHIMIE (FR) 1999-06-10 WO disclosed
WO-1998048628-A1 COMPOSITION FOR CONTROLLING HARMFUL BIO-ORGANISMS AND METHOD FOR CONTROLLING HARMFUL BIO-ORGANISMS USING THE SAME ISHIHARA SANGYO KAISHA, LTD. (JP) 1998-11-05 WO disclosed
EP-0298196-B1 IMIDAZOLE COMPOUNDS AND BIOCIDAL COMPOSITIONS COMPRISING THE SAME ISHIHARA SANGYO KAISHA, LTD. (JP) 1993-06-02 EP disclosed
US-4995898-A Imidazole compounds and biocidal composition comprising the same for controlling harmful organisms ISHIHARA SANGYO KAISHA, LTD. (JP) 1991-02-26 US disclosed
EP-0298196-A1 Imidazole compounds and biocidal compositions comprising the same ISHIHARA SANGYO KAISHA, LTD. (JP) 1989-01-11 EP disclosed