SCHEMBL9328936

SCHEMBL9328936

Nc1nc(Sc2ccccc2)nc2nc(-c3cccs3)nn12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 9/20 0.42
ADORA2B P29275 6/20 0.42
ADORA2A P29274 9/20 0.41
ADORA1 P30542 7/20 0.41
LMNA P02545 2/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
GLA P06280 1/20 0.36
GAA P10253 1/20 0.36
NPC1 O15118 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
HSD17B10 Q99714 1/20 0.36
CSNK1D P48730 1/20 0.34
TP53 P04637 1/20 0.34
MAPT P10636 1/20 0.34
FYN P06241 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9328560 0.85 ADORA3 (0.58) ADORA3ADORA2BADORA2AADORA1LMNA
SCHEMBL9327189 0.77 ADORA3 (0.61) ADORA3ADORA2BADORA2AADORA1ALDH1A1
SCHEMBL7828518 0.75 ADORA3 (0.73) ADORA3ADORA2BADORA2AADORA1
SCHEMBL9325713 0.74 ADORA3 (0.46) ADORA3ADORA2BADORA2AADORA1CSNK1D
SCHEMBL30596780 0.73 KDM4E (0.41) ADORA3ADORA2BADORA2AADORA1LMNA
SCHEMBL30596777 0.73 KDM4E (0.41) ADORA3ADORA2BADORA2AADORA1LMNA
SCHEMBL9325959 0.73 ADORA3 (0.48) ADORA3ADORA2BADORA2AADORA1
SCHEMBL9327033 0.73 ADORA3 (0.51) ADORA3ADORA2BADORA2AADORA1
SCHEMBL9328272 0.71 ADORA3 (0.47) ADORA3ADORA2BADORA2AKDM4ENPC1
SCHEMBL9429507 0.70 ADORA2A (0.66) ADORA3ADORA2BADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5356894-A Adenosine antagonists SYNGENTA LIMITED (GB) 1994-10-18 US disclosed
US-5270311-A [1,2,4]-Triazolo[1,5-a]and pyrazolo[2,3-a][1,3,5]triazine derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-12-14 US disclosed
EP-0459702-A1 Azole Derivatives ZENECA LIMITED (GB) 1991-12-04 EP disclosed