SCHEMBL932861

SCHEMBL932861

NC1=NCC2COCCC2(c2cccc(Br)c2)S1

nearest known ligand 0.33

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CHRNA1 P02708 1/20 0.32
CHRNG P07510 1/20 0.32
CHRNB1 P11230 1/20 0.32
CHRNB2 P17787 1/20 0.32
SLC6A2 P23975 1/20 0.32
CHRNB4 P30926 1/20 0.32
SLC6A4 P31645 1/20 0.32
CHRNA3 P32297 1/20 0.32
CHRNA4 P43681 1/20 0.32
SLC6A3 Q01959 1/20 0.32
CHRND Q07001 1/20 0.32
CTSD P07339 1/20 0.32
BACE1 P56817 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL934246 0.81 ALDH1A1 (0.34) CHRNA1CHRNGCHRNB1CHRNB2SLC6A2
SCHEMBL3691139 0.81 ALDH1A1 (0.34) CHRNA1CHRNGCHRNB1CHRNB2SLC6A2
SCHEMBL933050 0.76 HCRTR1 (0.37) BACE1
SCHEMBL932334 0.76 HCRTR1 (0.37) BACE1
Hydrochloric Acid SCHEMBL932779 0.74 BACE1 (0.54) CTSDBACE1
SCHEMBL6875209 0.73 BACE1 (0.48) BACE1
SCHEMBL14299100 0.73 BACE1 (0.48) BACE1
SCHEMBL933134 0.73 BACE1 (0.48) BACE1
SCHEMBL933387 0.72 USP2 (0.34)
SCHEMBL16418277 0.70 BACE1 (0.38) CHRNA1CHRNGCHRNB1CHRNB2SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2451793-A1 BACE INHIBITORS Eli Lilly and Company (US) 2012-05-16 EP disclosed
WO-2011005738-A1 BACE INHIBITORS ELI LILLY AND COMPANY (US) 2011-01-13 WO disclosed