SCHEMBL933050

SCHEMBL933050

CC(C)(C)OC(=O)NC1=NCC2COCCC2(c2cccc(Br)c2)S1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 1/20 0.37
HCRTR2 O43614 1/20 0.37
AAK1 Q2M2I8 3/20 0.35
USP30 Q70CQ3 2/20 0.33
BACE1 P56817 3/20 0.33
EGFR P00533 1/20 0.31
RAF1 P04049 1/20 0.31
KDR P35968 1/20 0.31
MAP2K2 P36507 1/20 0.31
MAP2K1 Q02750 1/20 0.31
AURKB Q96GD4 1/20 0.31
BCL2 P10415 1/20 0.31
BECN1 Q14457 1/20 0.31
FPR3 P25089 6/20 0.31
FPR2 P25090 6/20 0.31
BRD4 O60885 1/20 0.30
CREBBP Q92793 1/20 0.30
CTSB P07858 1/20 0.30
CTSS P25774 1/20 0.30
CTSK P43235 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL932334 1.00 HCRTR1 (0.37) HCRTR1HCRTR2AAK1USP30BACE1
SCHEMBL933488 0.90 HCRTR1 (0.37) HCRTR1HCRTR2AAK1BRD4CREBBP
SCHEMBL934246 0.86 ALDH1A1 (0.34)
SCHEMBL3691139 0.86 ALDH1A1 (0.34)
SCHEMBL932583 0.82 BACE1 (0.44) BACE1
SCHEMBL932781 0.80 BACE1 (0.32) AAK1BACE1
SCHEMBL966555 0.79 HCRTR1 (0.37) HCRTR1HCRTR2AAK1USP30BACE1
SCHEMBL6878525 0.79 HCRTR1 (0.37) HCRTR1HCRTR2AAK1USP30BACE1
SCHEMBL12851582 0.79 HCRTR1 (0.37) HCRTR1HCRTR2AAK1USP30BACE1
SCHEMBL967768 0.79 HCRTR1 (0.37) HCRTR1HCRTR2AAK1USP30BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011005738-A1 BACE INHIBITORS ELI LILLY AND COMPANY (US) 2011-01-13 WO disclosed