SCHEMBL934246

SCHEMBL934246

O=C(O)NC1=NCC2COCCC2(c2cccc(Br)c2)S1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.34
USP2 O75604 1/20 0.34
TSHR P16473 1/20 0.34
HSD17B10 Q99714 1/20 0.34
CHRNA1 P02708 1/20 0.32
CHRNG P07510 1/20 0.32
CHRNB1 P11230 1/20 0.32
CHRNB2 P17787 1/20 0.32
SLC6A2 P23975 1/20 0.32
CHRNB4 P30926 1/20 0.32
SLC6A4 P31645 1/20 0.32
CHRNA3 P32297 1/20 0.32
CHRNA4 P43681 1/20 0.32
SLC6A3 Q01959 1/20 0.32
CHRND Q07001 1/20 0.32
LMNA P02545 1/20 0.32
GAA P10253 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
HDAC1 Q13547 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3691139 1.00 ALDH1A1 (0.34) ALDH1A1USP2TSHRHSD17B10CHRNA1
SCHEMBL933387 0.88 USP2 (0.34) ALDH1A1USP2TSHRHSD17B10LMNA
SCHEMBL933050 0.86 HCRTR1 (0.37)
SCHEMBL932334 0.86 HCRTR1 (0.37)
SCHEMBL932861 0.81 CHRNA1 (0.32) CHRNA1CHRNGCHRNB1CHRNB2SLC6A2
SCHEMBL933478 0.80 BACE1 (0.47)
SCHEMBL968863 0.76 ALDH1A1 (0.34) ALDH1A1USP2TSHRHSD17B10CHRNA1
SCHEMBL968545 0.76 ALDH1A1 (0.34) ALDH1A1USP2TSHRHSD17B10CHRNA1
SCHEMBL16055857 0.71 ALDH1A1 (0.36) ALDH1A1CHRNA1CHRNGCHRNB1CHRNB2
SCHEMBL15321565 0.71 ALDH1A1 (0.36) ALDH1A1CHRNA1CHRNGCHRNB1CHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2451793-A1 BACE INHIBITORS Eli Lilly and Company (US) 2012-05-16 EP disclosed
WO-2011005738-A1 BACE INHIBITORS ELI LILLY AND COMPANY (US) 2011-01-13 WO disclosed