SCHEMBL9328769

SCHEMBL9328769

O=c1cc(-c2cccc(F)c2)oc2c(CBr)cccc12

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 9/20 0.63
CYP1A1 P04798 8/20 0.63
CYP1B1 Q16678 8/20 0.63
PRKDC P78527 1/20 0.63
GABRP O00591 7/20 0.59
GABRD O14764 7/20 0.59
GABRA1 P14867 7/20 0.59
GABRB1 P18505 7/20 0.59
GABRG2 P18507 7/20 0.59
GABRB3 P28472 7/20 0.59
GABRA5 P31644 7/20 0.59
GABRA3 P34903 7/20 0.59
GABRA2 P47869 7/20 0.59
GABRB2 P47870 7/20 0.59
GABRA4 P48169 7/20 0.59
GABRE P78334 7/20 0.59
GABRA6 Q16445 7/20 0.59
GABRG1 Q8N1C3 7/20 0.59
GABRG3 Q99928 7/20 0.59
GABRQ Q9UN88 7/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9329978 0.84 CYP1A2 (0.59) CYP1A2CYP1A1CYP1B1PRKDCGABRP
SCHEMBL9328614 0.84 CYP1A2 (0.59) CYP1A2CYP1A1CYP1B1PRKDCGABRP
SCHEMBL9328540 0.80 CYP1A1 (0.67) CYP1A2CYP1A1CYP1B1PRKDCGABRP
SCHEMBL31061033 0.77 CYP1A1 (1.00) CYP1A2CYP1A1CYP1B1PRKDCGABRP
SCHEMBL6617302 0.75 TERT (0.76) CYP1A2CYP1A1CYP1B1PRKDCGABRP
SCHEMBL8532 0.75 GABRP (1.00) CYP1A2CYP1A1CYP1B1PRKDCGABRP
SCHEMBL9327677 0.74 CYP2D6 (0.53) CYP1A2CYP1A1CYP1B1PRKDCGABRP
SCHEMBL9331009 0.74 AURKA (0.51) CYP1A2CYP1A1CYP1B1PRKDCGABRP
SCHEMBL29307653 0.73 CYP1A2 (0.63) CYP1A2CYP1A1CYP1B1PRKDCGABRP
SCHEMBL9160788 0.73 CYP1A2 (0.40) CYP1A2CYP1A1CYP1B1PRKDCCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0454728-B1 FLUORINATED FLAVONE ACETIC ACID UPJOHN CO (US) 1994-03-16 EP disclosed
US-5238954-A Antitumor agents THE UPJOHN COMPANY (US) 1993-08-24 US disclosed
EP-0454728-A1 FLUORINATED FLAVONE ACETIC ACID. UPJOHN CO (US) 1991-11-06 EP disclosed
WO-1990008143-A1 FLUORINATED FLAVONE ACETIC ACID THE UPJOHN COMPANY (US) 1990-07-26 WO disclosed