SCHEMBL9327677

SCHEMBL9327677

O=C(O)Cc1cccc2c(=O)cc(-c3cc(F)cc(F)c3)oc12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 3/20 0.53
CYP1A2 P05177 6/20 0.49
CYP3A4 P08684 3/20 0.49
CYP2C19 P33261 2/20 0.49
STAT6 P42226 1/20 0.49
CYP1A1 P04798 5/20 0.48
CYP1B1 Q16678 5/20 0.48
PRKDC P78527 2/20 0.48
GLA P06280 1/20 0.45
STING1 Q86WV6 1/20 0.45
XDH P47989 1/20 0.44
GABRP O00591 3/20 0.44
GABRD O14764 3/20 0.44
GABRA1 P14867 3/20 0.44
GABRB1 P18505 3/20 0.44
GABRG2 P18507 3/20 0.44
GABRB3 P28472 3/20 0.44
GABRA5 P31644 3/20 0.44
GABRA3 P34903 3/20 0.44
GABRA2 P47869 3/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9328614 0.91 CYP1A2 (0.59) CYP2D6CYP1A2CYP3A4CYP2C19STAT6
SCHEMBL9327900 0.90 CYP1A2 (0.56) CYP2D6CYP1A2CYP3A4CYP2C19STAT6
SCHEMBL9328729 0.89 CYP2D6 (0.49) CYP2D6CYP1A2CYP3A4CYP2C19STAT6
Mitoflaxone SCHEMBL106705 0.87 CYP1A2 (0.62) CYP2D6CYP1A2CYP3A4CYP2C19STAT6
SCHEMBL9328479 0.86 CYP2D6 (0.44) CYP2D6CYP1A2CYP3A4CYP2C19STAT6
SCHEMBL9327546 0.85 CYP1A2 (0.58) CYP2D6CYP1A2CYP3A4CYP2C19STAT6
SCHEMBL12835503 0.85 CYP1A2 (0.60) CYP2D6CYP1A2CYP3A4CYP2C19STAT6
SCHEMBL12835338 0.84 TDP1 (0.57) CYP2D6CYP1A2CYP3A4CYP2C19STAT6
SCHEMBL9327573 0.84 GLA (0.46) CYP2D6CYP1A2CYP3A4CYP2C19STAT6
SCHEMBL9328862 0.84 ALDH1A1 (0.51) CYP2D6CYP1A2CYP3A4CYP2C19STAT6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0454728-B1 FLUORINATED FLAVONE ACETIC ACID UPJOHN CO (US) 1994-03-16 EP claimed
US-5238954-A Antitumor agents THE UPJOHN COMPANY (US) 1993-08-24 US claimed
EP-0454728-A1 FLUORINATED FLAVONE ACETIC ACID. UPJOHN CO (US) 1991-11-06 EP claimed
WO-1990008143-A1 FLUORINATED FLAVONE ACETIC ACID THE UPJOHN COMPANY (US) 1990-07-26 WO claimed
EP-0454728-B1 FLUORINATED FLAVONE ACETIC ACID UPJOHN CO (US) 1994-03-16 EP disclosed
US-5238954-A Antitumor agents THE UPJOHN COMPANY (US) 1993-08-24 US disclosed
EP-0454728-A1 FLUORINATED FLAVONE ACETIC ACID. UPJOHN CO (US) 1991-11-06 EP disclosed
WO-1990008143-A1 FLUORINATED FLAVONE ACETIC ACID THE UPJOHN COMPANY (US) 1990-07-26 WO disclosed