SCHEMBL9329166

SCHEMBL9329166

Nc1nc(SC2CCCC2)nc2nc(-c3ccoc3)nn12

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 6/20 0.41
ADORA2B P29275 4/20 0.41
ADORA2A P29274 6/20 0.39
ADORA1 P30542 6/20 0.39
CSNK1D P48730 2/20 0.38
MEN1 O00255 1/20 0.33
USP2 O75604 1/20 0.33
ALDH1A1 P00352 1/20 0.33
TP53 P04637 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
ALOX15 P16050 1/20 0.33
KMT2A Q03164 1/20 0.33
HSD17B10 Q99714 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9325911 0.81 ADORA3 (0.62) ADORA3ADORA2BADORA2AADORA1
SCHEMBL9327392 0.80 ADORA3 (0.67) ADORA3ADORA2BADORA2AADORA1
SCHEMBL9325713 0.78 ADORA3 (0.46) ADORA3ADORA2BADORA2AADORA1CSNK1D
SCHEMBL9327228 0.76 ADORA2A (0.67) ADORA3ADORA2BADORA2AADORA1CSNK1D
SCHEMBL9328686 0.76 ADORA3 (0.42) ADORA3ADORA2BADORA2AADORA1CSNK1D
SCHEMBL23291366 0.69 ADORA2A (0.38) ADORA3ADORA2BADORA2AADORA1CSNK1D
SCHEMBL9328035 0.68 ADORA3 (0.66) ADORA3ADORA2BADORA2AADORA1CSNK1D
SCHEMBL23840696 0.62 ADORA3 (0.64) ADORA3ADORA2BADORA2AADORA1CSNK1D
SCHEMBL9328278 0.60 ADORA2A (0.60) ADORA3ADORA2BADORA2AADORA1ALDH1A1
SCHEMBL7145308 0.60 MAP3K5 (0.43) ADORA3ADORA2AADORA1MEN1USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5356894-A Adenosine antagonists SYNGENTA LIMITED (GB) 1994-10-18 US disclosed
US-5270311-A [1,2,4]-Triazolo[1,5-a]and pyrazolo[2,3-a][1,3,5]triazine derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-12-14 US disclosed
EP-0459702-A1 Azole Derivatives ZENECA LIMITED (GB) 1991-12-04 EP disclosed