SCHEMBL7145308

SCHEMBL7145308

Nc1cccc2nc(-c3ccoc3)nn12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP3K5 Q99683 1/20 0.43
AHR P35869 1/20 0.41
CYP11B2 P19099 1/20 0.38
ADORA3 P0DMS8 2/20 0.38
ADORA1 P30542 2/20 0.38
ADORA2A P29274 3/20 0.36
NUDT1 P36639 1/20 0.36
FYN P06241 2/20 0.34
MEN1 O00255 3/20 0.34
CYP1A2 P05177 3/20 0.34
CYP3A4 P08684 3/20 0.34
CYP2D6 P10635 3/20 0.34
KMT2A Q03164 3/20 0.34
CYP2C19 P33261 2/20 0.34
HSD17B10 Q99714 2/20 0.34
USP2 O75604 2/20 0.34
ALDH1A1 P00352 2/20 0.34
CLK4 Q9HAZ1 2/20 0.34
MAPT P10636 1/20 0.34
ALOX15 P16050 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7144401 0.79 ADORA3 (0.53) AHRCYP11B2ADORA3ADORA1ADORA2A
SCHEMBL7487566 0.78 KDM4E (0.40) AHRCYP11B2ADORA3ADORA1ADORA2A
SCHEMBL6863099 0.75 ADORA2A (0.45) MAP3K5ADORA3ADORA1ADORA2A
SCHEMBL7152951 0.74 ADORA2A (0.56) ADORA3ADORA1ADORA2A
SCHEMBL2772772 0.73 NUDT1 (0.65) MAP3K5ADORA1ADORA2ANUDT1FYN
SCHEMBL7151749 0.73 ALDH1A1 (0.49) CYP11B2ADORA3MEN1CYP1A2KMT2A
SCHEMBL6871806 0.72 ADORA2A (0.42) ADORA3ADORA1ADORA2A
SCHEMBL6869842 0.71 PLAU (0.48) MAP3K5ADORA2AMEN1KMT2AHSD17B10
SCHEMBL6869244 0.70 ADORA2A (0.67) ADORA2A
SCHEMBL6871623 0.69 ADORA2A (0.67) ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6506772-B1 Pharmaceutically active salts thereof with activity as adenosine receptor ligands are disclosed. These compounds are the adenosine receptor. HOFFMANN-LA ROCHE INC. 2003-01-14 US disclosed